Clozapine-d8是Clozapine的氘代同位素化合物。Clozapine 是一种抗精神病药物，具有高效结合多种神经受体的能力，广泛用于精神分裂症的研究。

Guanfacine HCl is a centrally acting antihypertensive with α2-adrenoceptor agonist with Kd value of 31 nM for α2A-adrenoceptor while displaying 60-fold selectivity over α2B-adrenoceptors, causing a decrease in heart rate and peripheral vascular resistance.

ST91是一种 α2-肾上腺素能受体 (α2AR) 激动剂，激活 α2AAR 和其他亚型，具有脊柱抗伤害作用。

Arotinolol is a blocker of both α- and β-receptor, and also acts as a β3 receptor agonist. It is used in the treatment of high blood pressure and essential tremor.

JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM.

Terazosin HCl is an α-adrenergic (AL-fa ad-ren-ER-jik) blocker used in the therapy of hypertension and benign prostatic hypertrophy with climination half-life‎ of ‎12 hours.

Detomidine HCl is an imidazole-derived α2-adrenergic agonist, used in veterinary medicine for sedation of large animals.

Tolazoline HCl is a competitive non-selective α-adrenergic receptor antagonist, used as a a vasodilator directly acting on blood vessels and also increasing cardiac output.

Brimonidine tartrate is an α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, used to treat glaucoma through a dual mechanism of action by reducing aqueous humor production and increasing uveoscleral outflow.

Nicergoline is a non-selective alpha-adrenergic receptor antagonist which can decrease vascular resistance and increase arterial blood flow in the brain, improving the utilization of oxygen and glucose by brain cells.

Medetomidine is an agonist of α2-adrenoceptor with Ki value of 1.08 nM, used as both a surgical anesthetic and analgesic.

Potent, selective 5-HT6 antagonist

Scopine HCl salt is a naturally occuring α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock and also s a potential brain-targeting moiety for enhancing the brain uptake efficiency of chlorambucil.

B-HT 920 is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity.

Rilmenidine Phosphate is an oxazole-derived agonist of adrenergic receptor α2 and Imidazoline receptor, used in trials studying the treatment of hypertension and chronic kidney disease.

Vibegron是一种有效的、选择性 β3-肾上腺素能受体激动剂 (EC₅₀=1.1 nM)，主要用于治疗膀胱过度活动症及严重急症尿失禁，具有显著的治疗效果。

Carazolol-d7是 Carazolol 的氘代同位素标记物，常用于药代动力学研究，帮助探究 Carazolol 的代谢途径。

Practolol是一种选择性 β1 肾上腺素能受体拮抗剂，可用于心律失常研究。

Romifidine是一种 α2 肾上腺素受体激动剂，表现出显著的镇静作用，广泛用于麻醉及疼痛管理，特别是在动物模型中的应用较为常见。

Meranzin, a natural product isolated and purified from the peel of Citrus maxima, can induce similar effect to Fructus Aurantii on intestinal motility and it was, at least in part, mediated by stimulation of H1 histamine receptors.