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货号 产品名 纯度
A846150 Vibegron

97%
A1229955 Carazolol-d7/(±)-卡拉洛尔-d7

98% 98%atom%D
A1213192 Clozapine-d8

cp98%, 98%D
A1061990 Romifidine hydrochloride

98%+
A1188867 JP1302

97%
A1154387 (Rac)-Rotigotine

97%
A436598 Guanfacine/胍法辛

Guanfacine is a selective α2A receptor agonist.

98%+
A810155 Guanfacine HCl/盐酸胍法辛

Guanfacine HCl is a centrally acting antihypertensive with α2-adrenoceptor agonist with Kd value of 31 nM for α2A-adrenoceptor while displaying 60-fold selectivity over α2B-adrenoceptors, causing a decrease in heart rate and peripheral vascular resistance.

99%
A1167355 (-)-Viloxazine HCl

(S)-Viloxazine Hydrochloride is the S-isomer of Viloxazine, a selective norepinephrine reuptake inhibitor (NRI) that can be used as an antidepressant.

99%+
A444012 Ritodrine HCl/盐酸利托君

Ritodrine HCl activates β-2 adrenergic receptor through binding to β-2 adrenergic receptors on outer membrane of myometrial cell, used to stop premature labor.

99+%
A1209339 ST91

97%
A1178877 SR59230A

SR59230A is a potent and selective Adrenergic Receptor β3 antagonist with IC50 values of 40, 408, and 648nM for Adrenergic Receptor β3, β1 and β2, respectively. It shows blood-brain barrier penetrability.

98%
A267563 Cadralazine

Cadralazine is an antihypertensive of the hydrazinophthalazine chemical class.

95%
A494835 DSP-4 HCl/DSP-4,肾上腺能神经毒素

DSP-4 showed neurotoxic effects on noradrenergic neurons of adult and developing rats.

99%+
A587683 Deserpidine/地舍平

Deserpidine is an antihypertensive drug related to reserpine which occurs naturally in Rauvolfia spp.

98%
A1678579 Golcadomide

98%
A316550 JP1302 2HCl

JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM.

99%+
A366659 AGN 192836

AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively.

99%+
A272742 Alfuzosin HCl/盐酸阿夫唑嗪

Alfuzosin HCl is an antagonist of α1 adrenergic receptor used to treat benign prostatic hyperplasia (BPH).

98%
A597542 Phentolamine HCl/盐酸苯酚胺

99%+
产品名 Adrenergic Receptor α-adrenergic receptor β-adrenergic receptor 其他靶点 纯度
Ivabradine HCl 98%
Maprotiline hydrochloride 98%
Cisatracurium besylate 98%
Yohimbine HCI 99+%
BMY 7378 ++

α1D-adrenoceptor, pKi: 5.1

α2C-adrenoceptor, pKi: 6.54

+

β1-adrenoceptor, pIC50: 5.1

97%
Asenapine maleate ++++

α2A-adrenergic receptor, pKi: 8.9

α2B-adrenergic receptor, pKi: 8.9

97%
Piribedil ++

adrenoceptor α2C, pKi: 7.2

adrenoceptor α2A, pKi: 7.1

98%
Prazosin HCl 95%
Silodosin 98%
Phenoxybenzamine HCl 98%
Naftopidil +++

α1D-adrenergic receptor, Ki: 20 nM

α1A-adrenergic receptor, Ki: 3.7 nM

98%
Naftopidil 2HCl +

α1-adrenergic receptor, IC50: 0.2 μM

97%
Alfuzosin HCl 98%
Terazosin HCl 99%
Atipamezole 95%
Phentolamine methanesulfonate salt 99%
Doxazosin mesylate 98%
Tolazoline HCl 98%
Zenidolol hydrochloride ++++

β1-adrenergic receptor, Ki: 611nM

β2-adrenergic receptor, Ki: 0.7nM

98%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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