Propafenone (SA-79) 是一种钠通道阻滞剂，具有抗心律失常作用。它还对β受体具有高亲和力（IC50=32 nM）。Propafenone通过诱导线粒体功能障碍和凋亡抑制食管癌增殖。

Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH 是一种抗肿瘤活性分子。

Dabuzalgron (Ro 115-1240)是一种口服活性的选择性α-1A肾上腺素受体激动剂，用于动物模型的尿失禁缓解。它通过维持线粒体功能来预防阿霉素诱导的心脏毒性。

Rotigotine 是一种有效的多巴胺受体激动剂，其对多巴胺D3受体的Ki值为0.71 nM，对D2、D5、D4受体的Ki值为4-15 nM，对多巴胺D1受体的Ki值为83 nM。Rotigotine 是5-HT1A受体的部分激动剂和α2B-肾上腺素受体的拮抗剂。Rotigotine 可用于帕金森病（PD）的研究。

Guanfacine is a selective α2A receptor agonist.

Guanfacine HCl is a centrally acting antihypertensive with α2-adrenoceptor agonist with Kd value of 31 nM for α2A-adrenoceptor while displaying 60-fold selectivity over α2B-adrenoceptors, causing a decrease in heart rate and peripheral vascular resistance.

Ritodrine HCl activates β-2 adrenergic receptor through binding to β-2 adrenergic receptors on outer membrane of myometrial cell, used to stop premature labor.

Terazosin is a selective alpha1-antagonist used for treatment of symptoms of benign prostatic hyperplasia (BPH).

Arotinolol is a blocker of both α- and β-receptor, and also acts as a β3 receptor agonist. It is used in the treatment of high blood pressure and essential tremor.

Cadralazine is an antihypertensive of the hydrazinophthalazine chemical class.

DSP-4 showed neurotoxic effects on noradrenergic neurons of adult and developing rats.

Deserpidine is an antihypertensive drug related to reserpine which occurs naturally in Rauvolfia spp.

JP 1302 dihydrochloride is an antagonist of α2C-adrenoceptor with Ki value of 28 nM.

Alfuzosin HCl is an antagonist of α1 adrenergic receptor used to treat benign prostatic hyperplasia (BPH).

L-765314 is a potent and selective α1b adrenergic receptor antagonist with Kis of 5.4±0.6 nM and 2.0±0.66 nM for rat and human α1b adrenergic receptor, respectively.