Cytotoxicity against human A549 cells, IC50=0.019 μM
21470864
human 786-O cells
Cytotoxic assay
72 h
Cytotoxicity against human 786-O cells after 72 hrs by MTT assay, IC50=0.022 μM
19637874
human A549 cells
Function assay
Antagonist activity at human PAR2 expressed in human A549 cells assessed as inhibition of 2f-LIGRLO-NH2-induced NFkappaB activation by luciferase reporter gene assay, IC50=0.014 μM
23895492
human A549 cells
Cytotoxic assay
72 h
Cytotoxicity against human A549 cells after 72 hrs by MTT assay, IC50=0.059 μM
19637874
human Bel7402 cells
Cytotoxic assay
72 h
Cytotoxicity against human Bel7402 cells after 72 hrs by MTT assay, IC50=0.02 μM
19637874
human DU145 cells
Cytotoxic assay
72 h
Cytotoxicity against human DU145 cells after 72 hrs by MTT assay, IC50=0.024 μM
19637874
human HCT116 cells
Cytotoxic assay
72 h
Cytotoxicity against human HCT116 cells after 72 hrs by MTT assay, IC50=0.01 μM
19637874
human HCT15 cells
Cytotoxic assay
72 h
Cytotoxicity against human HCT15 cells after 72 hrs by MTT assay, IC50=0.029 μM
19637874
human HeLa cells
Cytotoxic assay
72 h
Cytotoxicity against human HeLa cells after 72 hrs by MTT assay, IC50=0.047 μM
19637874
human HO8910 cells
Cytotoxic assay
72 h
Cytotoxicity against human HO8910 cells after 72 hrs by MTT assay, IC50=0.028 μM
19637874
human HT-29 cells
Cytotoxic assay
Cytotoxicity against human HT-29 cells, IC50=2.1 nM
21470864
human K562 cells
Cytotoxic assay
72 h
Cytotoxicity against human K562 cells after 72 hrs by MTT assay, IC50=0.05 μM
19637874
human KB cells
Cytotoxic assay
72 h
Cytotoxicity against human KB cells after 72 hrs by MTT assay, IC50=0.043 μM
19637874
human KBM5 cells
Cytotoxic assay
72 h
Cytotoxicity against imatinib-resistant human KBM5 cells harboring Bcr-Abl T315I mutant after 72 hrs by MTS assay, IC50=0.0083 μM
20149665
human MCF7 cells
Cytotoxic assay
72 h
Cytotoxicity against human MCF7 cells after 72 hrs by MTT assay, IC50=0.019 μM
19637874
human MDA-MB-231 cells
Cytotoxic assay
72 h
Cytotoxicity against human MDA-MB-231 cells after 72 hrs by MTT assay, IC50=0.024 μM
19637874
human MKN28 cells
Cytotoxic assay
72 h
Cytotoxicity against human MKN28 cells after 72 hrs by MTT assay, IC50=0.2 μM
19637874
human MOLT4 cells
Cytotoxic assay
72 h
Cytotoxicity against human MOLT4 cells after 72 hrs by MTT assay, IC50=0.017 μM
19637874
human PC3 cells
Proliferation assay
72 h
Antiproliferative activity against human PC3 cells after 72 hrs by SRB assay, IC50=0.02 μM
20833543
human Rh30 cells
Cytotoxic assay
72 h
Cytotoxicity against human Rh30 cells after 72 hrs by MTT assay, IC50=0.014 μM
19637874
human SGC7901 cells
Cytotoxic assay
72 h
Cytotoxicity against human SGC7901 cells after 72 hrs by MTT assay, IC50=0.015 μM
19637874
human SKOV3 cells
Cytotoxic assay
72 h
Cytotoxicity against human SKOV3 cells after 72 hrs by sulforhodamine B assay, IC50=0.006 μM
24378709
human SMMC7721 cells
Cytotoxic assay
72 h
Cytotoxicity against human SMMC7721 cells after 72 hrs by MTT assay, IC50=0.018 μM
19637874
human SW1116 cells
Cytotoxic assay
72 h
Cytotoxicity against human SW1116 cells after 72 hrs by MTT assay, IC50=0.052 μM
19637874
human U251 cells
Cytotoxic assay
Cytotoxicity against human U251 cells assessed as inhibition of cell proliferation by sulforhodamine B assay, IC50=0.033 μM
25467158
MDA-MB-468 cells
Cytotoxic assay
Cytotoxicity against human MDA-MB-468 cells by SRB assay, IC50=0.01 μM
19637874
MEF
Cytotoxic assay
72 h
Cytotoxicity against MEF after 72 hrs by MTS assay, IC5=9.2 μM
20149665
mouse 32D cells
Cytotoxic assay
72 h
Cytotoxicity against mouse 32D cells harboring wild type Bcr-Abl after 72 hrs by MTS assay, IC50=0.032 μM