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货号 产品名 纯度
A1155605 现货 ONC206

ONC206 是 ONC201 的类似物。ONC206 是一种选择性拮抗剂,对多巴胺 D2 类受体 (DRD2/3/4) 具有纳摩尔效力。ONC206 表现出广谱抗肿瘤活性。

97%
A185949 现货 BP 897 HCl

BP 897 hydrochloride是一种有效的部分多巴胺D3受体激动剂和弱D2受体拮抗剂。BP 897盐酸盐对多巴胺D3受体具有高亲和力(Ki=0.92 nM),对D2受体的亲和力是其的70倍(Ki=61 nM)。

98%
A1380175 现货 Tavapadon

Tavapadon (PF-06649751) 是一种口服活性、高选择性的多巴胺 D1/D5 受体部分激动剂。Tavapadon 有效促进运动和减少残疾,显示出治疗帕金森病的潜力。

97%
A306218 现货 Rotigotine/罗替戈汀

Rotigotine 是一种有效的多巴胺受体激动剂,其对多巴胺D3受体的Ki值为0.71 nM,对D2、D5、D4受体的Ki值为4-15 nM,对多巴胺D1受体的Ki值为83 nM。Rotigotine 是5-HT1A受体的部分激动剂和α2B-肾上腺素受体的拮抗剂。Rotigotine 可用于帕金森病(PD)的研究。

99%
A216412 现货 Tetramethylrhodamine Methyl Ester Perchlorate/四甲基若丹明甲酯酸铵

Tetramethylrhodamine Methyl Ester Perchlorate是膜可渗透的阳离子荧光探针,特异性识别线粒体膜电位,附着在线粒体上并产生明亮的荧光。在某些浓度下,罗丹明染料对细胞的毒性低,使其成为检测动物细胞、植物细胞和微生物线粒体的理想选择。

99%+
A1213192 现货 Clozapine-d8

cp98%, 98%D
A1177348 现货 (-)-GSK598809

95%
A1675522 现货 GBR-13069 2HCl

98%+
A585716 现货 Trimethobenzamide

95%
A1250019 现货 LY3154207

Y3154207 is a novel, potent, and subtype selective human D1 positive allosteric modulator (PAM) with minimal allosteric agonist activity (EC50 = 3 nM). In contrast to orthosteric agonists, LY3154207 showed a distinct pharmacological profile without a bell-shaped dose-response relationship or tachyphylaxis in preclinical models. Identification of a crystalline form of free LY3154207 from the discovery lots was not successful. Instead, a novel cocrystal form with superior solubility was discovered and determined to be suitable for development. LY3154207 is now in clinical development as a potential first-in-class D1 PAM for Lewy body dementia.

99%+
A819643 现货 GR 103691

GR 103691 is an effective and selective receptor antagonist of the dopamine D3 receptor (D3DR).

98+%
A747660 现货 Ro 10-5824 2HCl

Ro 10-5824 2HCl is an agonist of dopamine D4 receptor with Ki of 5.2 nM.

99%+
A764267 现货 Bromopride/溴必利

Bromopride is a dopamine antagonist with prokinetic properties, widely used as an antiemetic.

98%
A447591 现货 PD-168077 maleate

PD 168077 maleate is an agonist of D4 dopamine receptor with Ki of 8.7 nM. It can induce synaptic translocation of CaMK II to postsynaptic sites in cultured prefrontal cortical neurons.

98%+
A689993 现货 Dexpramipexole/右旋普拉克索

Dexpramipexole is a neuroprotective agent and weak non-ergoline dopamine agonist.

98%
A156825 现货 (+)-PD 128907 hydrochloride

(+)-PD 128,907 HCl is an agonist of D3 dopamine receptor with Ki of 2.3 nM.

98%
A1365603 现货 AZA1

98%+
A308996 现货 Pardoprunox HCl

Pardoprunox HCl is a partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist.

99%+
A1176487 现货 YM17E

98%+
A512636 现货 ABT-724 3HCl/ABT 724 三盐酸盐

ABT-724 3HCl is a potent and highly selective dopamine D4 receptor agonist with EC50s of 12.4 nM, 14.3 nM and 23.2 nM for human dopamine D4 receptor, rat D4 receptor and ferret D4 receptor.

97%
产品名 D1 receptor D2 receptor D3 receptor D4 receptor D5 receptor DAT Dopamine receptor 其他靶点 纯度
Penfluridol +

Dopamine receptor, Ki: 1.6 μM

98%
Ansofaxine HCl ++

Dopamine receptor, IC50: 491 nM

98%
Tetrahydroberberine,THB +

D2 receptor, pKi: 6.08

98+%
Prochlorperazine Maleate 95%
Olanzapine 99+%
Trifluoperazine ++++

Dopamine D2 receptor, IC50: 1.1 nM

98%
Ropinirole hydrochloride ++

D2 receptor, Ki: 29 nM

99%
Lurasidone ++++

D2 receptor, Ki: 1 nM

98%
Levosulpiride 99+%
Pridopidine 95%
Metoclopramide 99+%
Molindone HCl 98%
Sulpiride 99+%
Perospirone ++++

D2 receptor, Ki: 1.4 nM

99%
Perospirone HCl ++++

D2 receptor, Ki: 1.4 nM

98+%
Phenothiazine 98%
Pimozide +

Dopamine D1 receptor, Ki: 6600 nM

+++

Dopamine D2 receptor, Ki: 3.0 nM

++++

Dopamine D3 receptor, Ki: 0.83 nM

98%
Rotundine ++

D1 receptor, IC50: 166 nM

+

D2 receptor, IC50: 1.47 μM

+

D3 receptor, IC50: 3.25 μM

98%
Domperidone 99+%
ONC206 97%
Pimethixene maleate ++

Dopamine D1 Receptor, pKi: 6.37

+++

Dopamine D2 Receptor, pKi: 8.19

++

Dopamine D4.4 Receptor, pKi: 7.54

97%
Loxapine succinate ++

D2 receptor (Human), Ki: 62 nM

D1 receptor (human), Ki: 26 nM

++

D2 receptor (human), Ki: 24 nM

D2 receptor (bovine), Ki: 26 nM

+++

D4 receptor (human), Ki: 7.5 nM

99%
Chlorprothixene +++

D1 receptor, Ki: 18 nM

+++

D2 receptor, Ki: 2.96 nM

+++

D3 receptor, Ki: 4.56 nM

+++

D5 receptor, Ki: 9 nM

98%
SCH-23390 HCl ++++

D1 dopamine receptor, Ki: 0.2 nM

++++

D5 dopamine receptor, Ki: 0.3 nM

98%
MPP+ iodide 97%
σ1 Receptor antagonist-1 +

DAT, pKi: 5.8

97%
Benztropine mesylate ++

DAT, IC50: 118 nM

98%
Azaperone 98%
Ziprasidone HCl 98+%
Paliperidone 98%
Alizapride HCl 99+%
Amisulpride 98%
Quetiapine hemifumarate Adrenergic Receptor 98%
Clozapine N-oxide 99%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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