Clozapine-d8是Clozapine的氘代同位素化合物。Clozapine 是一种抗精神病药物，具有高效结合多种神经受体的能力，广泛用于精神分裂症的研究。

Tabernanthalog是一种5-HT2A 激动剂。在啮齿类动物中，Tabernanthalog 已被发现可促进结构神经可塑性并产生抗抑郁作用。

Temanogrel is a highly selective 5-HT2A receptor antagonist with Ki of 4.9 nM.

Lvguidingan is a potent anticonvulsant agent.

SB-242084 2HCl is a selective and brain-penetrant antagonist for the 5HT2C receptor.

SB 699551 is a selective 5-ht5a receptor antagonist (pKi values are 8.3, < 6.0, < 6.0, < 6.0, < 5.5 and < 5.5 for 5-ht5a, 5-HT1B/D, 5-HT2A, 5-HT2C, 5-HT1A and 5-HT7 receptors respectively).

5-HT2C/2B antagonist

(Z)-Thiothixene is serotonergic receptor antagonist.

ML 10302 HCl is a potent 5-HT4 partial agonist with EC50 of 4 nM.

Alverine Citrate is a 5-HT1A receptor antagonist with IC50 value of 101 nM.

Nefazodone HCl is a 5-HT2A receptor antagonist with Ki of 5.8 nM and an inhibitor of serotonin and noradrenalin uptake with IC50s of 290 and 300 nM respectively, it is an antidepressant drug.

Phenylbiguanide is a 5-HT3 receptor selective agonist with an EC50 of 3.0±0.1 μM.

Rizatriptan Benzoate is a triptan-class 5-HT1 receptor agonist, used to treat migraine headaches.

Pizotifen is a highly selective 5-HT receptor blocking agent, which is a benzocycloheptane based drug.

Amitriptyline HCl is a multiple-target molecular as an inhibitor of both 5-HT and NA reuptake (SNRI), and also a TrkA/B agonist.

Potent, selective 5-HT6 antagonist

PF-3084014 is a reversible inhibitor of γ-secretase with IC50 of 6.2 nM.

B-HT 920 is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity.

PNU-282987 free base是一种选择性 α7 乙酰胆碱受体(α7 nAChR)激动剂，具有改善认知功能的研究潜力。

Sarizotan (EMD 128130) is an orally active serotonin 5-HT1A receptor and dopamine receptor agonist. Sarizotan (EMD 128130) exhibits IC50 values of 6.5 nM (rat 5-HT1A), 0.1 nM (human 5-HT1A), 15.1 nM (rat D2), 17 nM (human D2), 6.8 nM (human D3) and 2.4 nM (human D4.2), respectively[1].