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货号 产品名 纯度
A884075 现货 GSK189254A

GSK189254A 是一种强效且选择性的组胺 H3 受体拮抗剂,人类和大鼠 H3 受体的 pKi 值分别为 9.59-9.90 和 8.51-9.17。

99%
A104244 现货 VUF10460

VUF10460 是一种非咪唑类组胺 H4 受体激动剂,对大鼠 H4 受体的结合具有 pKi 值为 7.46。

99%+
A148043 现货 Latrepirdine 2HCl/拉曲吡啶二盐酸盐

Latrepirdine dihydrochloride是一种神经活性化合物,对组胺能、α-肾上腺素能和 5-羟色胺能受体具有拮抗活性。Latrepirdine 刺激淀粉样前体蛋白 (APP) 的降解代谢和 β-淀粉样蛋白 (Aβ) 的分泌。

98%
A798995 现货 Betazole 2HCl

95+%
A1217678 现货 H4R antagonist 3

98%
A611587 现货 Buclizine/布克立嗪

97%
A202923 现货 Lodoxamide tromethamine

Lodoxamide tromethamine is used as an ophthalmic solution that specially applying to the eye.

99%+
A312159 现货 Brompheniramine maleate/马来酸溴苯那敏

Brompheniramine maleate is an antagonist of histamine H1 receptors.

98%
A370864 现货 Lodoxamide/洛草氨酸

Lodoxamide is an agonist of GPR35.

98%+
A114849 现货 Decloxizine/去氯羟嗪

Decloxizine is a histamine 1 receptor antagonist.

99%+
A653792 现货 Bavisant/巴维桑特

Bavisant is a highly selective, orally active antagonist of the human H3 receptor with a mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD.

99%
A642303 现货 S 38093

S 38093 is a brain-penetrant antagonist/inverse agonist of H3 receptors.

99%+
A147384 现货 Tripelennamine HCl/盐酸吡苄明

Tripelennamine HCl is an antagonist of H1-receptor that used as a psychoactive drug with antipruritic activity.

98%
A128330 现货 Mianserin hydrochloride/盐酸米安色林

Mianserin HCl is inverse agonist of H1 receptor and can be act as a psychoactive agent of the tetracyclic antidepressant.

99+%
A676591 现货 (R)-(-)-α-Methylhistamine 2HCl/(R)-(-)-α-甲基组胺二盐酸盐

95%
A156843 现货 Niaprazine/尼普拉嗪

95%
A825701 现货 Dimethindene

97%
A584050 现货 Roxatidine Acetate HCl/盐酸罗沙替丁醋酸酯

Roxatidine acetate HCl is a slective antagonist of histamin H2 receptor.

98%
A534590 现货 Ciproxifan maleate

Ciproxifan maleate is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes.

99%+
A313360 现货 Cetirizine/西替利嗪

Cetirizine, a second-generation antihistamine, is a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria.

99%+
产品名 H1 receptor H2 receptor H3 receptor H4 receptor Histamine receptor 其他靶点 纯度
Hydroxyzine 2HCl 99+%
Cyclizine 97%
Loratadine +

B(0)AT2, IC50: 4 μM

98%
Desloratadine ++

Histamine H1 receptor, IC50: 51 nM

98%
Doxylamine succinate 99%
Ebastine 98%
Tripelennamine HCl +

H1 receptor, IC50: 30 μM

98%
Meclizine dihydrochloride 98%
Chlorpheniramine maleate +++

Histamine H1 receptor, IC50: 12 nM

99%
Diphenhydramine HCl 99%
Alcaftadine ++++

H1 receptor, pKi: 8.5

++

H2 receptor, pKi: 7.2

98%+
Fexofenadine HCl ++

Histamine H1 receptor, IC50: 246 nM

99%+
Bilastine +++

H1 receptor, Ki: 44.15 nM

98%
Pemirolast potassium 98%
Bepotastine besilate +

Histamine H1 receptor, pIC50: 5.7

98%
Mizolastine +++

Histamine H1 receptor, IC50: 47 nM

98%
Brompheniramine maleate 98%
Carbinoxamine maleate salt 99+%
Clemastine fumarate ++++

Histamine H1 receptor, IC50: 3 nM

98%
Ketotifen fumarate salt 95%
Rupatadine Fumarate ++

Histamine H1 receptor, Ki: 102 nM

PAFR 98%
Famotidine 97%
Roxatidine Acetate HCl +

Histamine H2 receptor, IC50: 3.2 μM

98%
Lafutidine 99%
Cimetidine 98%
Nizatidine ++++

Histamine H2 receptor, IC50: 0.9 nM

AChE 98%
Ranitidine 99%
Betahistine +

Histamine H3 receptor, IC50: 1.9 μM

98%
Ciproxifan maleate +++

Histamine H3 receptor, IC50: 9.2 nM

99%+
S 38093 ++

rat H3 receptor, Ki: 1.44 μM

human H3 receptor, Ki: 1.2 μM

99%+
JNJ-7777120 ++++

Histamine H4 receptor, Ki: 4.5 nM

98%
Azelastine HCl 98%
Epinastine HCl 98%
Levodropropizine 97%
Cyproheptadine hydrochloride 98%
Hesperetin 97%
Olopatadine HCl 98%
Mianserin hydrochloride 99+%
Buclizine 2HCl 97%
Latrepirdine 2HCl GluR 98%
Cetirizine 2HCl 98%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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