Cav 2.2 blocker 1是一种 N 型钙离子通道 (Cav 2.2) 抑制剂，对疼痛研究具有重要应用。

VK-II-36是一种类 Carvedilol 的化合物，能够抑制肌浆网钙释放，抑制早期和延迟后去极化诱发的触发活动，适用于研究局灶性室性心律失常及相关心血管疾病的治疗。

SOICR-IN-1是一种 store-overload induced calcium release (SOICR) 抑制剂，IC₅₀ 为 14.6 μM。该化合物用于心律失常的研究，通过调节钙离子释放改善心脏功能。

Carboxyamidotriazole is a blocker of non-voltage dependent calcium channel with anti-inflammatory activity.

H-DL-o-Tyr-OH是一种苯丙氨酸的代谢物，作为形成儿茶酚胺的前体，被用作β-地中海贫血中蛋白质氧化损伤的生物标志物。。

Mibefradil 2HCl is calcium channel blocker with moderate selectivity for T-type Ca2+ channels displaying

TGR5 receptor agonist, a potent TGR5 (GPCR19) agonist, showed improved potency in the U2-OS cell assay (pEC50 = 6.8) and in melanophore cells (pEC50 = 7.5).

Strontium ranelate stimulates the calcium sensing receptors (CaSR) and leads to the differentiation of pre-osteoblast to osteoblast which increases the bone formation.

Ned 19是一种选择性的 NAADP 拮抗剂，具有膜透性，能够以非竞争性机制抑制 NAADP 介导的 Ca2+ 信号通路，IC₅₀ 为 65 nM。Ned 19 强烈抑制肿瘤生长、血管生成和肺转移，在抗癌领域具有广泛应用前景。

Hyperoside, a natural product isolated and purified from the herb of Hypericum perforatum L., with neuro-protective, anti-inflammatory and antioxidative effects, promotes ECV304 cell proliferation, may cause herb-drug interactions when co-administrated with CYP2D substrates and serve as a protective agent by alleviating microglia activation in disorders such as Parkinson's disease.

Neomycin Trisulfate Salt is an aminoglycoside antibiotic and calcium channel protein inhibitor.

Carbamazepine is a blocker of sodium channel with IC50 of 131 μM in rat brain synaptosomes. It is an anticonvulsant drug.

Mirogabalin besylate 是一种选择性的电压门控钙通道 α2δ 亚基的有效配体，对 α2δ-1 和 α2δ-2 的亲和力分别为 13.5 nM 和 22.7 nM。

YS-201是 一种二氢吡啶类钙通道拮抗剂，可用于心绞痛和高血压研究。

Methyl homoveratrate 是 RWJ-26240 的体内代谢物，可在血浆、尿液和粪便中检测到。McN5691 (RWJ-26240) 是一种电压依赖性钙通道阻滞剂。

Rhyncholphylline, an alkaloid isolated and purified from the herbs of Uncaria rhynchophylla., can protect against ischemic damage and glutamate-induced neuronal death, and also inhibit MA impairment in cultured neurons in vitro. Ca2+ channel blocker.

Praeruptorin E is a cardiotonic agent with selective cardiac calcium channel agonistic effect.

S107 is a RyR-selective 1,4-benzothiazepine derivative that stabilizes RyR2 channels by enhancing the binding affinity of calstabin2 to mutant and/or PKA-phosphorylated channels.

Heteroclitin D是一种从 Kadsura 药用植物中提取的木质素，具有抗脂质过氧化活性，并通过抑制 L 型钙离子通道调控钙离子流入，具有潜在的心血管保护作用。

ZSET1446 是一种新型的认知增强剂，可改善多种阿尔茨海默病模型中的学习障碍。