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货号 产品名 纯度
A1326789 10-Cl-BBQ

Aryl Hydrocarbon Receptor (AhR) Agonists, Signal Transduction Modulators

98%
A311620 CAY 10465

99%+
A922304 Brevifolincarboxylic acid/短叶苏木酚酸

99%+
A1209932 SGA360

97%
A1463321 Tapinarof/苯烯莫德

97%
A282299 GNF351

GNF351 is a full aryl hydrocarbon receptor (AHR) antagonist. GNF351 competes with a photoaffinity AHR ligand for binding to the AHR with IC50 of 62 nM.

99%+
A160463 D-Kynurenine/D-犬尿氨酸

99%+
A624664 L-Kynurenine sulfate

95%
A163287 ITE

ITE is an AhR agonist with Ki value of 3nM, and also inhibits TGF-β-induced human myofibroblast differentiation.

98%
A256874 Cardamonin/豆蔻明

Cardamonin (Cardamomin), a natural flavone isolated from Alpinia katsumadai Hayata, acts as an aryl hydrocarbon receptor (AhR) activator. Cardamonin alleviates inflammatory bowel disease by the inhibition of NLRP3 inflammasome activation via an AhR/Nrf2/NQO1 pathway .

97%
A186535 Galangin/高良姜素

Galangin functions as an antagonist of the aryl hydrocarbon receptor and also inhibits CYP1A1 (IC50 = 1 μM). It belongs to flavonoids and can be extracted from the rhizome of Zingiber officinale Roscoe with anti-inflammatory properties.

98+%
A135866 Indole-3-carbinol/3-吲哚甲醇

Indole-3-Carbinol is a naturally occuring plant hormone found in cruciferous vegetables, which can both inhibit carcinogenesis in several animal species and enhance tumor incidence if administered at a post-initiation stage.

98%
A310855 Benvitimod

Benvitimod is a non-steroidal anti-inflammatory drug (NSAID) potentially for the treatment of atopic dermatitis.

98%
A204811 Formononetin/刺芒柄花素

Formononetin can act as an agonist of aryl hydrocarbon receptor (EC50 = 130 nM) and has prevention of breast cancer, prostate cancer and colon cancer. Formononetin could be extracted from the bark of Ononis natrix L..

98+%
A639949 Potassium 1H-indol-3-yl sulfate/吲苷钾盐

98%
A1209574 MeBIO

98%+
A898906 PDM11

PDM 11 is a derivative of the antioxidant trans-resveratrol.

99%+
A108671 StemRegenin 1

StemRegenin 1 is an AhR antagonist with IC50 of 127 nM. Also, it stimulates the proliferation and differentiation of CD34+ hematopoietic progenitor cells.

99%+
A1000372 Phortress

Aryl Hydrocarbon Receptor (AhR) Agonists, Signal Transduction Modulators

97%
A525118 CH-223191

CH-223191 is a ligand-selective antagonist of the Ah (Dioxin) receptor.

99%+
产品名 AhR 其他靶点 纯度
StemRegenin 1 ++

Aryl hydrocarbon receptor (AhR), IC50: 127 nM

99%+
CH-223191 +++

AhR, IC50: 30 nM

99%+
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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