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货号 产品名 纯度
A1176847 HC-070

98%
A1176676 TC-I 2014

99%+
A1164188 TRPM8-IN-1

98%
A990716 M8-B

99%+
A1365324 TRPM4-IN-1

99%+
A1512658 Moringin/辣木籽素

99%+
A1601979 (1R,2R)-ML-SI3

99%+
A266033 Vanillyl alcohol/4-羟基-3-甲氧基苄醇

Vanillyl alcohol is a free radical scavenger with anticonvulsive and bile secretion promoting effect. It can be extracted from the herbs of Gastrodia elata Bl..

95%
A658572 A-967079

A 967079 is a selective TRPA1 channel blocker (IC50 values are 67 and 289 nM at human and rat TRPA1 receptors respectively).

98%
A209665 Chembridge-5861528

Chembridge-5861528 is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-evoked calcium influx (IC50 values are 14.3 and 18.7μM respectively).

99%+
A224797 BCTC

BCTC is a potent and specific inhibitor of transient receptor potential cation channel subfamily M member 8 (TRPM8) in prostate cancer (PCa) DU145 cells.

99%+
A666937 Hydroxy-α-sanshool/羟基-α-山椒素

99%+
A208947 (Z)-Capsaicin/(Z)-辣椒素

Zucapsaicin is a synthetic cis isomer of natural capsaicin that has therapeutic efficacy in pain accompanying osteoarthritis of the knee.

95%
A1176853 TRPM8 antagonist 2

TRPM8 antagonist 14 is a tryptophan-derived selective TRPM8 antagonist with IC50 value of 0.2nM. It showed significant target coverage in both an icilin-induced WDS (at 1-30 mg/kg s.c.) and oxaliplatin-induced cold allodynia (at 0.1-1 μg s.c.) mice models.

98%+
A433794 SAR7334

SAR7334 is a potent TRPC6 (Transient receptor potential cation channel, subfamily C, member 6) inhibitor.

99+%
A757208 Pyr10

Pyr 10 is a TRPC3-selective inhibitor. IC50 of Ca2+ influx inhibition by Pyr10 in carbachol-stimulated YFP-TRPC3-transfected HEK293 cells for ROCE and thapsigargin-depleted native RBL-2H3 cells for SOCE is 0.72 uM and 13.08 uM.

99%+
A510332 Pyr6

Pyr6 is a selective inhibitor of TRPC3 with IC50 of 0.49 μM (Ca2+ influx inhibition in thapsigargin depleted native RBL-2H3 cells).

98%+
A892019 GSK2193874

GSK2193874 is a selective transient receptor potential vanilloid 4 (TRPV4) blocker with IC50 value of 0.04 μM.

99%+
A231850 RQ-00203078

RQ-00203078 is a selective antagonist of TRPM8 with IC50 of 8.3 nM.

99%+
A835423 ML204/4-甲基-2-(1-哌啶基)-喹啉

ML204 is a selective antagonist of TRPC4 ion channel with IC50 of 0.96 μM and 2.6 μM in fluorescent and electrophysiological assays respectively.

99%+
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