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PKC 相关产品
PKC 亚型比较

全部(211) Modulator(1) Antagonist(1) Inhibitor(23) Activator(4)

货号			产品名	纯度
A102655	现货	促	Pinoresinol diMethyl ether/松脂素二甲醚	97%
A1193875	现货	促	Bisindolylmaleimide III	99%+
A279706	现货	促	Darovasertib LXS196 is a potent and orally active protein kinase C (PKC) inhibitor used for the treatment of uveal melanoma.	99%+
A1177150	现货	促	p32 Inhibitor M36	99%+
A1598854	现货	促	WAY-301398	99%+
A911160	现货	促	Ingenol Mebutate/巨大戟醇甲基丁烯酸酯 Ingenol Mebutate 是大戟属 (Euphorbia peplus) 的活性成分和 PKC 的调节剂，对 PKC-α、PKC-β、PKC-γ、PKC-δ 和 PKC-ε 的 Ki 值分别为 0.3、0.105、0.162、0.376 和 0.171 nM。	98%
A905085	现货	促	Daphnoretin Daphnoretin (Dephnoretin) 是从Wikstroemia indica中提取的，具有抗病毒活性。Daphnoretin 通过直接激活蛋白激酶 C（类似于 PMA），从而激活 NADPH 氧化酶。	98%
A1806341	现货	促	PKC-theta inhibitor hcl	99%+
A2192875	现货	促	CWI1-2 HCl	98%
A701829	现货	促	R59949	99%+
A1363185	现货	促	PKC-iota inhibitor 1 PKC-iota inhibitor 1 PKC-ι ℩ inhibitor with IC50 value of 0.34μM.	99%+
A429214	现货	促	Aurothiomalate sodium/金硫丁二钠	99%+
A909799	现货	促	Decursin/紫花前胡素 Decursin ((+)-Decursin) 是一种有效的抗癌剂，具有细胞毒性和强效激活蛋白激酶 C (PKC) 的作用。Decursin 诱导细胞凋亡和 G1 期细胞周期停滞。Decursin 在 48 小时内减少 CDK2、CDK4、CDK6 和 cyclin D1 蛋白的表达。Decursin 抑制细胞增殖和迁移，具有抗肿瘤、抗炎和镇痛活性。	99%+
A238262	现货	促	Protein kinase inhibitor H-7 2HCl	99%+
A1210826	现货	促	ML192	97%
A200976	现货	促	TAS-301 TAS-301 is an inhibitor of smooth muscle cell migration and proliferation, inhibits intimal thickening after balloon injury to rat carotid arteries.	99%+
A703737	现货	促	Hypericin/金丝桃素 Hypericin, a natural product isolated and purified from the herb of Hypericum perforatum L., is a photosensitive antiviral with anticancer and antidepressant agent derived from Hypericum perforatum.	99%+
A1210808	现货	促	MitoPQ	97%
A1159144	现货	促	Bisindolylmaleimide X HCl Bisindolylmaleimide xHCl is a potent protein kinase C (PKC) inhibitor.	99%+
A122227	现货	促	Bisindolylmaleimide IV/双辛基马来酰亚胺 IV Bisindolylmaleimide IV is an inhibitor of protein kinase C.	97%

产品名	PKC ↓ ↑	PKCα ↓ ↑	PKCβ ↓ ↑	PKCγ ↓ ↑	PKCδ ↓ ↑	PKCε ↓ ↑	PKCζ ↓ ↑	PKCη ↓ ↑	PKCθ ↓ ↑	其他靶点	纯度
Daphnetin	+ PKC, IC50: 25.01 μM									EGFR,PKA	95%
Dequalinium Chloride											99%+
Quercetin	✔									Sirtuin,Src	97%
Myricetrin		✔									96%
Go 6983		+++ PKCα, IC50: 7 nM	+++ PKCβ, IC50: 7 nM	+++ PKCγ, IC50: 6 nM	+++ PKCδ, IC50: 10 nM		++ PKCζ, IC50: 60 nM				99%+
Go6976	+++ PKC, IC50: 7.9 nM	++++ PKCα, IC50: 2.3 nM	+++ PKCβ1, IC50: 6.2 nM							FLT3	99%+
Bisindolylmaleimide I		+++ PKCα, IC50: 20 nM	+++ PKCβ2, IC50: 16 nM PKCβ1, IC50: 17 nM	+++ PKCγ, IC50: 20 nM							99%+
Lawsone methyl ether			✔								99%
Sotrastaurin		++++ PKCα, Ki: 0.95 nM	++++ PKCβ1, Ki: 0.64 nM		++++ PKCδ, Ki: 2.1 nM	++++ PKCε, Ki: 3.2 nM		++++ PKCη, Ki: 1.8 nM	++++ PKCθ, Ki: 0.22 nM		99%+
Enzastaurin		++ PKCα, IC50: 39 nM	+++ PKCβ, IC50: 6 nM	+ PKCγ, IC50: 83 nM		+ PKCε, IC50: 110 nM					98%
Midostaurin		++ PKCα, IC50: 22 nM	++ PKCβ2, IC50: 31 nM PKCβ1, IC50: 30 nM	++ PKCγ, IC50: 24 nM	+ PKCδ, IC50: 330 nM	+ PKCε, IC50: 1.25 μM		+ PKCη, IC50: 160 nM			99%
Ro 31-8220 mesylate		++++ PKCα, IC50: 5 nM	+++ PKCβ2, IC50: 14 nM PKCβ1, IC50: 24 nM	++ PKCγ, IC50: 27 nM		++ PKCε, IC50: 24 nM					99%+
Staurosporine		++++ PKCα, IC50: 2 nM		++++ PKCγ, IC50: 5 nM	+++ PKCδ, IC50: 20 nM	++ PKCε, IC50: 73 nM		++++ PKCη, IC50: 4 nM			99%+
Ruboxistaurin HCl		+ PKCα, IC50: 0.36 μM	++++ PKCβ2, IC50: 5.9 nM PKCβ1, IC50: 4.7 nM	+ PKCγ, IC50: 0.3 μM	+ PKCδ, IC50: 0.25 μM			++ PKCη, IC50: 0.052 μM			99%+
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多，抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用，但抑制强度暂时没有相关数据。

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