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货号 产品名 纯度
A1006566 RCGD423

RCGD423 is a gp130 modulator, which prevents articular cartilage degeneration and promotes repair.

97%
A178453 Dofequidar

Dofequidar is a quinoline compound, which can reverse P-glycoprotein (P-gp)-mediated MDR.

98%
A670924 GP130 receptor agonist-1

gp130-agonist-2 is a brain penetrant gp130 agonist which protects against NMDA-induced toxicity and increases STAT3 phosphorylation.

99%+
A265225 Isosinensetin/异橙黄酮

Isosinensetin exhibits HIV-1 protease inhibiting and antioxidant activities. It is a natural product isolated and purified from the fruit of Citrus aurantium L..

99%+
A397520 Chrysosplenetin/猫眼草黄素

Chrysosplenetin, a natural product isolated and purified from the herbs of Laggera pterodonta, is a metabolic inhibitor of artemisinin.

98%
A356248 Sinapine thiocyanate/芥子碱硫氰酸盐

Sinapine, an alkaloid isolated and purified from the seeds of Raphanus sativus L., possess antioxidant and radio-protective activities, downregulats multi-drug resistance 1 (MDR1) expression.

99%+
A536549 Sinapine/芥子碱

Sinapine 是从十字花科种子中分离出来的生物碱,具有抗炎、抗氧化、抗肿瘤、抗血管生成和放射保护活性。它也是乙酰胆碱酯酶AChE)抑制剂,可用于研究阿尔茨海默病、共济失调、重症肌无力和帕金森病。

99%+
A658719 Encequidar

HM30181 is a potent and selective inhibitor of P-glycoprotein.

95+%
A351095 Elacridar/依克立达

Elacridar is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules.

99%+
A251517 Tariquidar/他立喹达

Tariquidar is a potent and selective noncompetitive inhibitor of P-glycoprotein with Kd of 5.1 nM, reverses drug resistance in MDR cell Lines.

99%+
A272992 Zosuquidar 3HCl/唑喹达三盐酸盐

Zosuquidar 3HCl is the 3HCl form of Zosuquidar. Zosuquidar is P-gp modulator that inhibited Pgp-ATPase activity 50-60% at 2 and 10μM and had no effect at 0.08 and 0.4μM.

99%+
A458424 Schisandrin/五味子醇甲

Schizandrin is a natural product possessing antioxidant and anti-inflammatory activities.

98%
A1176616 Reversan

97%
A1177698 MCI826

99+%
A1176545 P-gp inhibitor 1

A1176952 P-gp modulator 1

A1176445 TTT-28

99+%
A1210798 MC70

97%
A1210885 PGP-4008

97%
A1210921 Reversin 121

97%
产品名 P-gp 其他靶点 纯度
Elacridar BCRP 99%+
Zosuquidar 3HCl ++

P-gp, Ki: 60 nM

99%+
SC144 99%+
Tariquidar +++

P-gp, Kd: 5.1 nM

99%+
Schizandrin B 98%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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