Elacridar是一种口服活性 P-糖蛋白 (Pgp) 和乳腺癌耐药蛋白 (BCRP) 抑制剂，用于研究外排转运蛋白对药物在脑中分布的影响，并用于癌症研究。

Zosuquidar 3HCl(LY335979) 三盐酸盐是一种P-糖蛋白（P-gp）抑制剂，Ki值为59 nM。它具有抗肿瘤活性，可用于急性髓性白血病（AML）的研究。

Sinapine 是从十字花科种子中分离出来的生物碱，具有抗炎、抗氧化、抗肿瘤、抗血管生成和放射保护活性。它也是乙酰胆碱酯酶（AChE）抑制剂，可用于研究阿尔茨海默病、共济失调、重症肌无力和帕金森病。

RCGD423 is a gp130 modulator, which prevents articular cartilage degeneration and promotes repair.

Dofequidar is a quinoline compound, which can reverse P-glycoprotein (P-gp)-mediated MDR.

gp130-agonist-2 is a brain penetrant gp130 agonist which protects against NMDA-induced toxicity and increases STAT3 phosphorylation.

Sinapine, an alkaloid isolated and purified from the seeds of Raphanus sativus L., possess antioxidant and radio-protective activities, downregulats multi-drug resistance 1 (MDR1) expression.

HM30181 is a potent and selective inhibitor of P-glycoprotein.

Tariquidar is a potent and selective noncompetitive inhibitor of P-glycoprotein with Kd of 5.1 nM, reverses drug resistance in MDR cell Lines.

Schizandrin is a natural product possessing antioxidant and anti-inflammatory activities.

Chrysosplenetin, a natural product isolated and purified from the herbs of Laggera pterodonta, is a metabolic inhibitor of artemisinin.

Isosinensetin exhibits HIV-1 protease inhibiting and antioxidant activities. It is a natural product isolated and purified from the fruit of Citrus aurantium L..