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货号 产品名 纯度
A318812 MSDC 0160/米格列酮

MSDC-0160 is a prototype mTOR-modulating insulin sensitizer being studied to treat diabetes and Alzheimer's disease.

99%+
A330186 Rhoifolin/野漆树苷

Rhoifolin, a natural product isolated and purified from the leaves of Turpinia arguya Seem, hows monolithic proliferation inhibitory activities against Hela, A549 and MCF-7 cell lines, and may be beneficial for diabetic complications through their enhanced adiponectin secretion, tyrosine phosphorylation of insulin receptor-β and GLUT4. It was found to efficiently block the enzymatic activity of SARS-CoV 3CLpro.

99%+
A224689 Kaempferitrin/山奈苷

Kaempferitrin can activate insulin signaling pathway, phosphorylate Akt kinase and exert the transloocation of GLUT4, thus has antitumor, antidepressant and antidiabetic effects. Kaempferitrin is a natural product isolated and purified from the root of Kaempferia galangal L..

95%
A899724 Tolazamide/甲磺氮草脲

Tolazamide is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity.

99%+
A126440 Ceritinib/色瑞替尼

Ceritinib is potent inhibitor against ALK with IC50 of 0.2 nM, shows 40- and 35-fold selectivity against IGF-1R and InsR, respectively.

98%
A361478 BMS-536924

BMS-536924 is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM.

98%
A139562 Linsitinib

Linsitinib is highly potent, orally efficacious and highly selective, dual ATP-competitive inhibitor of IGF-1R (IC50= 35 nM) and insulin receptor (IC50=75 nM).

99%+
A462988 NVP-AEW541

NVP-AEW541 is a potent inhibitor of IGF-1R with IC50 of 86 nM, 27-fold greater selectivity for IGF-1R than InsR.

99%+
A135758 Cinnamic acid/肉桂酸,只含反式

Cinnamic acid can stimulate insulin secretion and improve glucose tolerance.

98% only trans
A184967 BMS-754807

BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.8 nM/1.7 nM, less potent to Met, Aurora A/B, TrkA/B and Ron, and shows little activity to Flt3, Lck, MK2, PKA, PKC etc.

99%+
A1163884 GIP, human/抑胃肽

Gastric Inhibitory Peptide (GIP), human is thought to act as an inhibitor of gastric functions. It also affects lipid metabolism and displays mitogenic and antiapoptotic effects in pancreatic β-cells.

99%
A1209494 HNMPA

97%
A1209951 HNMPA-(AM)3

97%
A1256703 (Pro3) GIP, human

98+%
A1256512 GIP (1-30) amide,human

A1256666 GIP (3-42), human

A1250513 S961

98%
A1250512 S961 TFA

98%
A1484668 Gastric Inhibitory Peptide, porcine

98+%
A1500064 DA-JC4

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