Bedaquiline, a diarylquinoline antibiotic that targets ATP synthase, is effective for the treatment of Mycobacterium tuberculosis infections.

Oligomycin A, a mitochondrial ATP synthase inhibitor, is isolated from Streptomyces species, exhibits anti-tumor and antibiotic activity.

BTB06584 is an IF1-dependent selective inhibitor of the mitochondrial F1Fo-ATPase.

Bedaquiline fumarate, a diarylquinoline antibiotic that targets ATP synthase, is effective for the treatment of Mycobacterium tuberculosis infections.

Bz 423 is an ATP synthase inhibitor woth IC50 ~5 μM.

Oligomycin Complex is a mixture of oligomycins A, B, and C. Oligomycin A is a selective inhibitor of mitochondrial F1FO-ATP synthase that induces apoptosis in a variety of cell types. Oligomycin B is a nonselective inhibitor of ATP synthases. Oligomycin B can reduce the rate of ATP depletion in myocardial ischemia and decrease calcium-induced calcium release oscillation frequency of rat sensory neurons.