GS-6201（CVT-6883）是一种选择性的腺苷A2B受体拮抗剂，对人类腺苷A2B受体具有高亲和力和选择性（Ki=22 nM）。

N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.

Tozadenant is a selective adenosine A2A receptor antagonist with Ki values of 11.5 nM on human A2A and 6 nM on rhesus A2A, which can improve motor function in animal models of Parkinson's disease.

Preladenant is a highly selective and competitive A2A receptor antagonist with Ki value of 1.1nM, used in trials studying the treatment of brain diseases, such as parkinson disease, movement disorders, antipsychotic agents and parkinsonian disorders.

BAY 2416964 is an antagonist of aryl hydrocarbon receptor (AhR) with IC50 of 341 nM.

Taminadenant is an antagonist of adenosine receptor.

CGS 15943 is a potent adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively.

AZD4635 is an A2AR antagonist which can reverse adenosine mediated T cell suppression.

N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM).

N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor, with Ki of 29 nM for rat ecto-5′-nucleotidase.

Alloxazine is a selective antagonist of A2B adenosine receptor.

N6-[2-(4-Aminophenyl)ethyl]adenosine is a potent, non-selective A3 adenosine receptor agonist.

BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.

Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.

Acefylline is an adenosine receptor antagonist, a stimulant drug of the xanthine chemical class.