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货号 产品名 纯度
A1953407 PSB-1901

98%+
A178913 N6-(2-Hydroxyethyl)adenosine/N6-(2-羟乙基)腺苷

N-(2-Hydroxyethyl)adenosine has been studied as an anticonvulsant through the activation of adenosine A1 receptor (AA1R). It attenuates cell death induced by H2O2 through antioxidant action.

96%
A100067 Tozadenant

Tozadenant is a selective adenosine A2A receptor antagonist with Ki values of 11.5 nM on human A2A and 6 nM on rhesus A2A, which can improve motor function in animal models of Parkinson's disease.

98+%
A120930 Preladenant

Preladenant is a highly selective and competitive A2A receptor antagonist with Ki value of 1.1nM, used in trials studying the treatment of brain diseases, such as parkinson disease, movement disorders, antipsychotic agents and parkinsonian disorders.

99%+
A1257495 BAY 2416964

BAY 2416964 is an antagonist of aryl hydrocarbon receptor (AhR) with IC50 of 341 nM.

99%+
A232307 Taminadenant

Taminadenant is an antagonist of adenosine receptor.

97%
A592542 Imaradenant

AZD4635 is an A2AR antagonist which can reverse adenosine mediated T cell suppression.

99%+
A598514 N6-Cyclohexyladenosine

N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM).

99%+
A1508915 VCP171

95%
A858213 N6-Benzyladenosine/N6-苄基腺苷

98%
A818008 BAY 60-6583

BAY 60-6583 is a potent adenosine A2B receptor agonist with EC50 of 2.83 nM for murine A2B receptor.

99%+
A791038 Istradefylline/伊曲茶碱

Istradefylline is a very potent, selective and orally active adenosine A2A receptor antagonist (Ki=2.2 nM) in experimental models of Parkinson's disease.

98%
A215378 Norisoboldine/去甲异波尔定

Norisoboldine is an isoquinoline alkaloid isolated and purfied from the roots of Lindera aggregata, which acts as an AhR agonist, and enhances the function of the adenosine A1 receptor.

98%
A520792 7-(2,3-Dihydroxypropyl)theophylline/二羟丙茶碱

Dyphylline, a xanthine derivative, acts as an adenosine receptor antagonist and phosphodiesterase inhibitor, which is used in the treatment of respiratory disorders.

98%
A325694 Proxyphylline/羟丙茶碱

Proxyphylline is a xanthine-derivatived antagonists of A1 and A2 adenosine receptors, which relaxe smooth muscles, particularly bronchial muscles.

99%
A229005 Theophylline-7-acetic Acid/茶碱乙酸

Acefylline is an adenosine receptor antagonist, a stimulant drug of the xanthine chemical class.

99+%
A724057 A2A receptor antagonist 1

99%+
A1501762 MIPS521

95%
A300603 1,3,9-Trimethylxanthine

97%
A155723 Vipadenant

Vipadenant is an adenosine antagonist with Ki of 1.3 nM and 68 nM for A2A and A1, respectively. Vipadenant is a selective A2A receptor antagonist with Ki values of 1.3, 68, 63, and 1,005 nM for A2A, A1, A2B, and A3 receptors, respectively, used in development for for Parkinson's disease.

99%+
产品名 Adenosine Receptor 其他靶点 纯度
ZM241385 99%+
Istradefylline +++

Adenosine A2A receptor, Ki: 2.2 nM

98%
Reversine +

human A3 adenosine receptor, Ki: 0.66 μM

98%
SCH58261 ++++

bovine A2a, Ki: 2.0 nM

rat A2a, Ki: 2.3 nM

99%+
A2A receptor antagonist 1 ++

A1R, Ki: 264 nM

A2AR, Ki: 4 nM

99%+
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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