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货号 产品名 纯度
A1324875 CH6953755

CH6953755 is a selective inhibitor of YES1 kinase with IC50 of 1.8 nM.

98%+
A230809 AMG-47a

AMG-47a is a Lck inhibitor that can decrease T cell proliferation with anti-inflammatory activity.

99%+
A146866 PP2

PP2 is a ATP-competitive inhibitor of the Src family of protein tyrosine kinases. The IC50s for p56lck, p59fynT, Hck, Src are 4 nM, 5 nM, 5 nM, 100 nM, respectively.

98%
A135851 WH-4-023

WH-4-023 is an inhibitor of Lck and Src with IC50 of 2 nM, 6 nM, respectively.

99%+
A724479 RK-24466

RK-24466 is an inhibitor of Lck (64-509) and LckCD isoforms with IC50s of <2 nM.

99%+
A1598758 HPK1-IN-2

95%
A523201 Src Inhibitor 1

Src inhibitor 1 is an inhibitor of Src and Lck with IC50 of 44 nM and 88nM.

99%
A1539742 Chrysotoxine

98%+
A1229415 HIV-IN-6

98%+
A1258085 Hck-IN-1

Hck Blocker compound B9 is a Nef-dependent Hck blocker with IC50 value of 2.8μM for Nef-Hck complex but >20μM for Hck alone. It binds directly to Nef via a pocket formed by the Nef dimerization interface and disrupts Nef dimerization in cells.

98%+
A742025 SU6656/2,3-二氢-N,N-二甲基-2-氧代-3-[(4,5,6,7-四氢-1H-吲哚-2-基)亚甲基] -1H-吲哚-5-磺酰胺

SU 6656 is an inhibitor of Src kinases and can target Src, Yes, Lyn, and Fyn with IC50 of 280 nM, 20 nM, 130 nM, 170 nM, respectively.

99%+
A1362232 DGY-06-116

DGY-06-116 is an irreversible covalent and selective Src inhibitor.

99%+
A259165 β-Hydroxyisovalerylshikonin/β-羟基异戊酰基紫草素

95%
A459806 PD-089828

99%+
A1328087 SI-2 HCl

SI-2 hydrochloride (EPH 116 hydrochloride) is a highly promising SRC-3 SMI: SRC-3 inhibitor (PPI), with IC50 values of 3-20 nM for breast cancer cell death. SI-2 hydrochloride (EPH 116 hydrochloride) has a much improved toxicity and pharmacokinetic profile, with acceptable oral availability[1].

99%+
A1602853 NCGC00262650

99%+
A1176814 eCF506

99%+
A333356 Bosutinib hydrate

95%
A769419 KX1-004

KX1-004 is a potent small molecule inhibitor of Src-PTK as a potential protective drug for NIHL.

97%
A161457 Tirbanibulin/特班布林

KX2-391 is an inhibitor of Src with IC50 of 9 nM-60 nM in cancer cells. It is the first clinical and peptidomimetic class Src inhibitor.

99%+
产品名 Fyn Lck Lyn Src Yes 其他靶点 纯度
Saracatinib ++

Fyn, IC50: 10 nM

++++

LCK, IC50: <4 nM

+++

Lyn, IC50: 5 nM

++++

c-Src, IC50: 2.7 nM

99%+
SU6656 +

Fyn, IC50: 170 nM

+

Lyn, IC50: 130 nM

+

Src, IC50: 280 nM

++

YES, IC50: 20 nM

99%+
PP1 +++

Fyn, IC50: 6 nM

+++

LCK, IC50: 5 nM

EGFR 99%+
PP2 +++

Fyn, IC50: 5 nM

++++

LCK, IC50: 4 nM

98%
WH-4-023 ++++

Lck, IC50: 2 nM

+++

Src, IC50: 6 nM

99%+
NVP-BHG 712 +

c-Src, IC50: 1.266 μM

99%+
CCT196969 ++

LCK, IC50: 0.02 μM

+

Src, IC50: 0.03 μM

98%
MNS +

Src, IC50: 29.3 μM

Syk,p97 98%
Tirbanibulin ++

Src (Hep 3B), GI50: 26 nM

Src (HuH7), GI50: 13 nM

99%+
PP121 ++

Src, IC50: 14 nM

VEGFR,PDGFR 99%+
Bosutinib ++++

Src, IC50: 1.2 nM

99%
Dasatinib monohydrate ++++

Src, IC50: 0.8 nM

98%
Quercetin PKC,Sirtuin 97%
Dasatinib ++++

Src, IC50: 0.8 nM

98%
Repotrectinib +++

Src, IC50: 5.3 nM

99%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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