 
        
        
        Maohuoside A是一种从淫羊藿(Epimedium brevicornu Maxim)根部提取的天然产物,通过 BMP 和 MAPK 信号通路促进大鼠间充质干细胞和骨髓来源的间充质干细胞的骨生成。
 
                                 
                                
                            

| 规格 | 价格 | 会员价 | 库存 | 数量 | |||
|---|---|---|---|---|---|---|---|
| {[ item.pr_size ]} | {[ getRatePriceInt(item.pr_rmb, 1,1) ]}{[ getRatePriceInt(item.pr_rmb_sale, 1,1) ]} {[ suihuo_tips(item.pr_tag_price, item.pr_am) ]} | {[ getRatePriceInt(item.pr_rmb, 1,1) ]}{[ getRatePriceInt(item.pr_rmb,item.pr_rate,1) ]} {[ suihuo_tips(item.pr_tag_price, item.pr_am) ]} | {[ getRatePriceInt(item.pr_rmb, 1,1) ]}{[ suihuo_tips(item.pr_tag_price, item.pr_am) ]} | {[ getRatePrice(item.pr_rmb_sale, 1,1,item.mem_isinteger) ]} {[ getRatePrice(item.pr_rmb,item.pr_rate,item.mem_rate,item.mem_isinteger) ]} {[ getRatePrice(item.pr_rmb,1,item.mem_rate,item.mem_isinteger) ]} | 现货 | 1周 咨询 | - + | 
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| 产品名称 | ALK1 ↓ ↑ | ALK2 ↓ ↑ | ALK3 ↓ ↑ | ALK4 ↓ ↑ | ALK6 ↓ ↑ | Smad3 ↓ ↑ | TGF-β ↓ ↑ | TGFβRI/ALK5 ↓ ↑ | TGFβRII ↓ ↑ | 其他靶点 | 纯度 | ||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| LDN193189 | ++++ ALK1, IC50: 0.8 nM | ++++ ALK2, IC50: 0.8 nM | +++ ALK3, IC50: 5.3 nM | +++ ALK6, IC50: 16.7 nM | 99%+ | ||||||||||||||
| LDN-212854 | ++++ ALK1, IC50: 2.4 nM | ++++ ALK2, IC50: 1.3 nM | + ALK3, IC50: 85.8 nM | + ALK4, IC50: 2133 nM | + ALK5, IC50: 9276 nM | 99%+ | |||||||||||||
| ML347 | ++ ALK1, IC50: 46 nM | ++ ALK2, IC50: 32 nM | 98% | ||||||||||||||||
| K02288 | ++++ ALK1, IC50: 1.8 nM | ++++ ALK2, IC50: 1.1 nM | ++ ALK3, IC50: 34.4 nM | +++ ALK6, IC50: 6.4 nM | 99%+ | ||||||||||||||
| LDN-193189 2HCl | ++++ ALK1, IC50: 0.8 nM | ++++ ALK2, IC50: 0.8 nM | +++ ALK3, IC50: 5.3 nM | +++ ALK6, IC50: 16.7 nM | 99% | ||||||||||||||
| LDN-214117 | ++ ALK2, IC50: 24 nM | 98% | |||||||||||||||||
| DMH-1 | + ALK2, IC50: 107.9 nM | 99%+ | |||||||||||||||||
| SB-505124 | + ALK4, IC50: 129 nM | ++ ALK5, IC50: 47 nM | 99%+ | ||||||||||||||||
| Vactosertib | +++ ALK4, IC50: 13 nM | +++ ALK5, IC50: 11 nM | 99%+ | ||||||||||||||||
| Alantolactone | ✔ | 98% | |||||||||||||||||
| (E/Z)-SIS3 free base | ✔ | 97% | |||||||||||||||||
| Pirfenidone | ✔ | 98% | |||||||||||||||||
| Hesperetin | ✔ | 97% | |||||||||||||||||
| RepSox | ++++ TGFβR1(ALK5), IC50: 4 nM | 98% | |||||||||||||||||
| GW788388 | +++ ALK5, IC50: 18 nM | 98% | |||||||||||||||||
| LY364947 | ++ TGFβRI, IC50: 59 nM | + TGFβRII, IC50: 0.4 μM | 98% | ||||||||||||||||
| SD-208 | ++ TGF-βRI (ALK5), IC50: 48 nM | 99% | |||||||||||||||||
| SB-525334 | +++ TGFβR1(ALK5), IC50: 14.3 nM | 99%+ | |||||||||||||||||
| LY2109761 | ++ TβRI, Ki: 38 nM | + TβRII, Ki: 300 nM | 99%+ | ||||||||||||||||
| Galunisertib | ++ TβRI, IC50: 56 nM | 98% | |||||||||||||||||
| SB 431542 | + ALK5, IC50: 94 nM | 99%+ | |||||||||||||||||
| 1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。 | |||||||||||||||||||
| 描述 | Maohuoside A, a natural product isolated and purified from the roots of Epimedium brevicornu Maxim, seems to enhance the osteogenesis of rMSC and bone marrow-derived mesenchymal stem cells at least partly via the BMP and MAPK signaling pathways and bone morphogenetic protein signalling, respectively. | 
| 计算器 | ||||
| 存储液制备 |  | 1mg | 5mg | 10mg | 
| 1 mM 5 mM 10 mM | 1.82mL 0.36mL 0.18mL | 9.12mL 1.82mL 0.91mL | 18.23mL 3.65mL 1.82mL | |
| CAS号 | 128988-55-6 | 
| 分子式 | C27H32O12 | 
| 分子量 | 548.54 | 
| SMILES Code | O=C1C(O)=C(C2=CC=C(OC)C=C2)OC3=C(CCC(C)(O)C)C(O[C@H]4[C@@H]([C@H]([C@@H]([C@@H](CO)O4)O)O)O)=CC(O)=C13 | 
| MDL No. | MFCD31697553 | 
| 别名 | |
| 运输 | 蓝冰 | 
| InChI Key | KKZRHUJZVYWXFJ-RGLOOMPQSA-N | 
| Pubchem ID | 14583586 | 
| 存储条件 | In solvent -20°C: 3-6个月 -80°C: 12个月 Pure form Keep in dark place, sealed in dry, 2-8°C | 
| 溶解方案 | 请根据您的动物给药指南选择适当的溶解方案。 以下溶解方案都请先按照体外实验的方式配制澄清的储备液,再依次添加助溶剂: ——为保证实验结果的可靠性,澄清的储备液可以根据储存条件,适当保存;体内实验的工作液,建议现用现配,当天使用; 以下溶剂前显示的百分比是指该溶剂在终溶液中的体积占比;如在配制过程中出现沉淀、析出现象,可以通过加热和/或超声的方式助溶 
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