Ambeed.cn

首页 / 抑制剂/激动剂 / / PKG

货号 产品名 纯度
A274191 现货 PKG drug G1

PKG Drug G1 targets C42 of PKG Iα. PKG drug G1 can couple to vasodilation and blood pressure lowering by a C42 PKG Iα-independent mechanism.

99%+
A193859 现货 Fasudil HCl/盐酸法舒地尔

Fasudil HCl (HA-1077; AT877)是一种非特异性RhoA/ROCK抑制剂,同时抑制蛋白激酶,对ROCK1的Ki为0.33 μM,对ROCK2PKAPKCPKGIC50值分别为0.158 μM、4.58 μM、12.30 μM和1.650 μM。Fasudil盐酸盐还是一种强效的Ca2+通道拮抗剂和血管扩张剂。

98%
A171227 现货 H-89 2HCl

H-89 2HCl是一种高效且选择性的蛋白激酶A(PKA)抑制剂,IC50为48 nM,对PKGPKC和酪蛋白激酶的抑制作用较弱。

99%+
A914568 现货 HA-100/HA 100二盐酸盐

HA-100 is an inhibitor of cGMP-dependent protein kinase (PKG), cAMP-dependent protein kinase (PKA), protein kinase C (PKC) and MLC-kinase (IC50 values are 4, 8, 12 and 240 μM, respectively).

97%
A2422082 SMA4

98%
A185330 HA-100 2HCl

HA-100 is an isoquinoline compound with an added piperazinylsulfonyl group that acts as an inhibitor of protein kinases (PKs), including PKA, PKC, and PKG (IC50s = 8, 12, and 4 µM, respectively).

98%
A555108 PKG inhibitor peptide

97%
A1158556 KT5823

KT 5823 is a selective inhibitor of the cGMP-dependent protein kinase (PKG) (Ki values are 0.23, 4 and > 10 μM for inhibition of PKG, PKC and PKA respectively). KT 5823 inhibits SNP-stimulated PKG activity with an IC50 of 60 nM in dispersed smooth muscle cells and has little effect on PKA activity at concentrations of up to 10 μM.

98%
A2420832 PKG1α activator 3

98%
A2792206 PKG drug G1

99%
A2791295 H-89 2HCl

99%
A2792816 HA-100/HA 100二盐酸盐

99%
Ambeed 相关网站 Ambeed.cn Ambeed.com
Ambeed
关于我们
联系我们
资讯中心
网站地图
产品手册
  • 批次文件查询
  • 客户支持
    技术支持
    专业术语
    缩略词释义
    质量手册
    产品咨询
    计算器
    活动政策
    订购方法
    积分商城
    活动声明
    联系我们
    400-920-2911 sales@ambeed.cn tech@ambeed.cn
    Ambeed 只为有资质的科研机构、医药企业基于科学研究或药证申报的用途提供医药研发服务,不为任何个人或者非科研性质用途提供服务。