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货号 产品名 纯度
A1209771 AZ10606120 2HCl

AZ10606120 dihydrochloride is a selective, high affinity antagonist for P2X7 receptor (P2X7R) at human and rat with an IC50 of ~10 nM. AZ10606120 dihydrochloride is little or no effect at other P2XR subtypes. AZ10606120 dihydrochloride has anti-depressant effects and reduces tumour growth .

99%+
A270115 A-804598

A-804598 is a competitive, and selective P2X7 receptor antagonist with IC50 of 10 nM, 9 nM and 11 nM in rat, mouse and human P2X7 receptors respectively.

99%+
A451786 AF-353

AF-353 is a potent and orally bioavailable P2X3/P2X2/3 receptor antagonist, inhibits human and rat P2X3 (pIC50= 8.0).

99%+
A628940 A 438079

A 438079 is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line).

99%+
A1167270 RO-3

RO-3 is a selective homomeric P2X3 and heteromeric P2X2/3 receptor antagonist.

98%+
A720722 JNJ-47965567

JNJ 47965567 is a potent and selective P2X7 antagonist (pIC50 values are 8.3, 7.5 and 7.2 for human, mouse and rat receptors respectively).

99%+
A111744 Cytidine-5'-triphosphate disodium salt dihydrate/三磷酸胞苷二钠

CTP Disodium Dihydrate is a P2X4 purinergic receptor agonist.

97%
A357468 Oxatomide/欧诗美锭

Oxatomide is a first-generation antihistamine of the diphenylmethylpiperazine (benzhydrylpiperazine) class.

99%+
A455366 KN-62

KN-62 is a selective and potent inhibitor of calmodulin-dependent protein kinase II (CaMK-II) with IC50 of 0.9 μM, KN-62 also displays noncompetitive antagonism at P2X7 receptors in HEK293 cells, with an IC50 value of approximately 15 nM..

98%
A1364936 BAY-1797

99%+
A585229 Gardenoside/羟异栀子苷

Gardenoside, a natural product isolated and purified from the fruits of Gardenia jasminoides Ellis, has anti-inflammatory, analgesic activities.

99%+
A152651 A 438079 HCl

A 438079 HCl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line).

99%+
A497149 A-317491

A-317491 is a potent and selective non-nucleotide antagonist of P2X3 and P2X2/3 receptors with Ki values of 22 nM and 9 nM for human P2X3 and P2X2/3 receptors.

99%+
A503454 Gefapixant

Gefapixant is an orally active P2X3 receptor (P2X3R) antagonist with IC50s of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors.

98%
A1226351 BX430

BX430 is selective P2X4 allosteric antagonist with IC50 of 0.54 μM.

99%+
A985017 AZ 11645373

95%
A1209443 NF110

97%
A1209318 TC-P 262

97%
A1211018 α,β-Methylene ATP trisodium

99+%
A1209292 Ro 0437626

97%
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