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货号 产品名 纯度
A1807773 现货 GW406108X(Z/E)

GW406108X(Z/E)是一种具有生物活性的化合物,主要作为Kif15(Kinesin-12)的特异性抑制剂。它还显示出对ULK1(Unc-51 like kinase 1)的ATP竞争性抑制作用,

98%
A647852 现货 Litronesib

Litronesib is a selective, allosteric inhibitor of Eg5, which may result in mitotic disruption, apoptosis and consequently cell death in tumor cells that are actively dividing.

98%
A231503 现货 GSK-923295

GSK-923295 是一种特异性的着丝粒相关蛋白 E (CENP-E) 驱动蛋白 ATP 酶活性的变构抑制剂,对人和犬的 Ki 值分别为 3.2±0.2 nM 和 1.6±0.1 nM。

99%+
A654863 现货 SB-743921 HCl

SB-743921 is a potent KIF11 inhibitor with Ki value of 0.1 nM.

99%+
A1152213 现货 Filanesib hydrochloride/ARRY-520盐酸盐

Filanesib hydrochloride是一种 Kinesin spindle protein (KSP) 抑制剂,能够干扰细胞分裂。它在癌症治疗中展现出显著的抗增生活性。

99%
A101991 现货 Monastrol

Monastrol is a specific and allosteric inhibitor of mitotic molecular motor kinesin Eg5 with IC50 value of 14 μM.

98%
A154438 现货 BRD9876

BRD9876 is a selective inhibitor of MM1S growth. It is selective for microtubule bound Eg5 and causes a rapid arrest in G2/M phase.

95%
A279561 现货 Ispinesib/伊斯平斯

Ispinesib is a quinazolinone-derived, specific and reversible kinesin spindle protein inhibitor with Kiapp value of 1.7 nM.

99%+
A174095 现货 AZ3146

AZ3146 is a selective and potent Mps1 inhibitor with IC50 value of 35 nM.

98+%
A519540 现货 MPI-0479605

MPI-0479605 is a potent and selective ATP competitive Mps1 with IC50 value of 1.8 nM.

99%+
A106724 现货 H-Cys(Trt)-OH/S-三苯甲基-L-半胱氨酸

H-Cys(Trt)-OH is a potent and selective inhibitor of mitotic kinesin Eg5 with IC50 value of 140 nM.

95%
A187476 现货 Dimethylenastron

Dimethylenastron is specific and reversible mitotic motor kinesin Eg5 inhibitor with IC50 value of 200 nM.

99%+
A394288 现货 K858 (Racemic)

K858 is a selective and ATP-uncompetitive mitotic kinesin Eg5 inhibitor with IC50 value of 1.3 μM.

98%
A719211 现货 CW-069

CW069 is a selective and allosteric microtubule motor protein HSET inhibitor with IC50 value of 75 μM.

99%+
A1176954 Eg5 Inhibitor V, trans-24

A1353331 SR31527 chloride

97%
A1399086 PVZB1194

98%
A724767 EMD534085

98%
A1356160 SB-743921 free base

98%
A1604020 KSP-IA

98%
产品名 Kinesin 其他靶点 纯度
SB-743921 HCl ++++

KSP (P388 cells), IC50: 14.4 nM

KSP, Ki: 0.07 nM

99%+
GSK-923295 ++

CENP-E, Ki: 3.2 nM

99%+
Ispinesib +++

KSP (HsEg5), Ki app: 1.7 nM

99%+
AZ3146 +

Mps1, IC50: ~35 nM

98+%
MPI-0479605 ++

Mps1, IC50: 1.8 nM

99%+
BAY1217389 +++

Mps1, IC50: 0.63 nM

98%
ARQ 621 98%
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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