Cyclo(RGDyK) is a highly potent and selective inhibitor for the αvβ3 integrin with a IC50 of 0.94 nM.

Leukadherin-1 is allosteric activator of CD11b/CD18 with EC50 value of 4 μM for increasing CD11b/CD18-dependent cell adhesion to fibrinogen.

Surfactin C1 是一种两亲性生物表面活性剂。Surfactin C1 抑制白血病细胞 (HL-60) 与人脐静脉内皮细胞 (HUVEC) 之间的粘附，抑制 ICAM-1 和 VCAM-1 等粘附分子的表达。

BTT-3033 是一种口服活性、构象选择性的 α2β1 抑制剂（EC50: 130 nM），可结合 α2I 结构域。BTT-3033 抑制血小板与 I 型胶原的结合和细胞增殖，并诱导凋亡。BTT-3033 可用于前列腺癌、炎症和心血管疾病的研究。

GLPG 0187 is a potent αv integrin inhibitor with IC50 values of 1.2-3.7 nM. It inhibits osteoclastic bone resorption and angiogenesis in vitro and in vivo. Also it suppresses epithelial-mesenchymal transition (EMT) and migration of PC-3M-Pro4/luc cells, without inhibiting cell growth.

A-205804 是一种口服活性、强效、选择性的 E-selectin 和 ICAM-1 表达抑制剂，IC50 值分别为 20 nM 和 25 nM，可用于慢性炎症性疾病的研究。

Cilengitide TFA是一种高效且选择性的整合素抑制剂，对 αvβ3 和 αvβ5 受体的 IC50 分别为 4 nM 和 79 nM。

Tirofiban is a non-peptide reversible antagonist of the platelet integrin glycoprotein (GP) IIb/IIIa receptor used as an antiplatelet drug.

TR-14035 is a dual antagonist of both integrin α4β7 and integrin α4β1 with IC50 values of 7 nM and 87 nM, respectively, used as an anti-inflammatory agent.

Arg-Gly-Asp is a cell adhesion motif which can mimic cell adhesion proteins and bind to integrins.

Cyclo(-RGDfK) is a potent and selective inhibitor of the αvβ3 integrin.

RGD 肽 (GRGDNP) 是一种整合素-配体相互作用抑制剂，通过竞争性抑制 α5β1 与细胞外基质（ECM）的结合起作用。RGD 肽 (GRGDNP) 通过增强促胱氨酸酶-3 活化和自加工的构象变化促进凋亡。在细胞粘附、迁移、生长和分化中起着关键作用。