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货号 产品名 纯度
A902254 现货 Telotristat etiprate/特罗司他马尿酸盐

Telotristat etiprate (LX1606 Hippurate) 是一种色氨酸羟化酶抑制剂,能减少血清素的产生。

99%+
A439308 现货 LX-1031

LX1031 is an oral, small molecule tryptophan 5-hydroxylase (TPH) inhibitor that reduces serotonin(5-HT) synthesis peripherally.

98%
A855563 现货 Telotristat ethyl

LX1606 is an orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.

99%+
A927595 现货 Ro 61-8048

Ro 61-8048 is an inhibitor of kynurenine 3-hydroxylase which can potently and competitively inhibit kynurenine 3-monooxygenase with Ki value and IC50 value of 4.8 nM and 37 nM, respectively.

99%+
A148106 现货 Nepicastat HCl

Nepicastat HCl is a potent and selective dopamine β-hydroxylase (DBH) inhibitor with IC50 value of 9 nM.

98%
A564408 现货 p-Ethynylphenylalanine

98%+
A400559 现货 Vitexin/牡荆素

Vitexin exhibits inhibition of carbohydrate hydrolase with IC50 of 244 μM and shows antioxidant activity in DPPH bleaching assay (IC50 = 24.2 μM). It is an apigenin flavone c-glycosidea isolated and purified from the seeds of Vitex trifolia L. with antinociceptive, antimyeloperoxidase, and anti-inflammatory activities.

98% HPLC
A701042 现货 Sapropterin 2HCl/盐酸沙丙蝶呤

Sapropterin 2HCl is a synthetic form of BH4 that is approved for the treatment of BH4 responsive PKU.

99%+
A744554 现货 Uric acid/尿酸

Uric acid activates NFκB in a variety of cell culture models including proximal tubular cells. Uric acid suppresses 1-α hydroxylase mRNA and protein expression in dose dependent and time dependent manner.

98%
A724867 现货 LP-533401

LP-533401 is an inhibitor of Tryptophan hydroxylase 1.

98%+
A148184 现货 Tetrahydropapaverine HCl/四氢罂粟碱盐酸盐

Tetrahydropapaverine HCl is a papaverine-derived inhibitor of TPH with the IC50 value of 5.7 μM.

97%
A624425 现货 H-α-Me-Tyr-OH/α-甲基-L-酪氨酸

Metyrosine is a selective tyrosine hydroxylase enzyme inhibitor. Metyrosine exerts anti-inflammatory and anti-ulcerative effects. Metyrosine significantly inhibits high COX-2 activity. Metyrosine is a very effective agent for blood pressure control.

95%
A129937 现货 H-HoArg-OH/高精氨酸

H-HoArg-OH (L-Homoarginine) is an organ-specific, uncompetitive inhibitor of human liver and bone alkaline phosphohydrolases.

97%
A256716 现货 H-DL-α-Me-Tyr-OH/α-甲基-DL-酪氨酸

97%
A867181 α-Methyltyrosine methyl ester HCl/α-甲基-DL-酪氨酸甲酯盐酸盐

98%
A349635 Scabertopin/地胆草内酯

Scabertopin, a natural product isolated and purified from the herbs of Elephantopus scaber Linn., exhibits significant antitumor effect in vitro in a concentration-dependent manner.

98+%
A1150650 GSK 366

97%
A617374 ACT-678689

97%
A529761 UPF-648

UPF-648 is a potent kynurenine 3-monooxygenase (KMO) inhibitor, exhibits highly active at 1 μM(81 ± 10% KMO inhibition), and is ineffective at blocking KAT activity.

99+%
A658929 LP-533401 HCl/LP-533401盐酸盐

LP-533401 HCl is an inhibitor of Tryptophan hydroxylase 1.

97%
产品名 Hydroxylase 其他靶点 纯度
Ro 61-8048 +++

KMO, Ki: 4.8 nM

KMO, IC50: 37 nM

99%+
DMOG 98%
Nepicastat HCl +++

Human dopamine-beta-hydroxylase, IC50: 9 nM

Bovine dopamine-beta-hydroxylase, IC50: 8.5 nM

98%
Telotristat etiprate 99%+
1. 鼠标悬停在“+”上可以显示相关IC50的具体数值。"+"越多,抑制作用越强。2. "✔"表示该化合物对相应的亚型有抑制作用,但抑制强度暂时没有相关数据。
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