Ambeed.cn

首页 / 抑制剂/激动剂 / / SRPK

货号 产品名 纯度
A476468 现货 ML281

ML281 是一种强效、选择性的喹喔啉基 STK33 抑制剂,IC50 值为 14 nM。

99%+
A1149118 现货 GSK8612

GSK8612是一种高度选择性和高效的Tank结合激酶-1(TBK1)抑制剂,对重组TBK1的pIC50为6.8。

99%+
A297057 现货 Midostaurin/米哚妥林

Midostaurin (PKC412; CGP 41251) 是一种口服活性、可逆的多靶点蛋白激酶抑制剂,抑制PKCα/β/γ、Syk、Flk-1、AktPKAc-Kit、c-Fgr、c-SrcFLT3PDGFRβ和VEGFR1/2的IC50值范围为22到500 nM。它还上调内皮一氧化氮合酶(eNOS)基因表达,并表现出强大的抗癌作用。

99%
A460722 现货 4μ8C

4μ8C(IRE1抑制剂III)是一种靶向IRE1α的小分子抑制剂。

99%+
A517820 现货 Sotrastaurin

Sotrastaurin (AEB071) 是一种高效且口服活性的泛 PKC 抑制剂,对 PKCθ、PKCβ、PKCα、PKCη、PKCδ PKCε 的 Ki 值分别为 0.22 nM、0.64 nM、0.95 nM、1.8 nM、2.1 nM 和 3.2 nM。

99%+
A333732 现货 Chelerythrine Chloride/盐酸白屈菜红碱

Chelerythrine Chloride是一种强效、细胞渗透的蛋白激酶C抑制剂,IC50为660 nM。此外,它抑制Bcl-XL-Bak BH3肽的结合,IC50为1.5 μM,并将Bax从Bcl-XL中置换出来。Chelerythrine Chloride诱导凋亡自噬

99%
A814222 现货 ILK-IN-2

ILK-IN-1 is an ILK inhibitor with IC50 of 0.6 μM.

98%+
A361136 现货 WNK463

WNK463 is a potant With-No-Lysine (WNK) kinase inhibitor with IC50s of 5/1/6/9 nM for WNK1/2/3/4.

98%
A1327308 现货 ILK-IN-3

ILK-IN-3 is an integrin linked kinase inhibitor.

99%+
A1263609 现货 Netarsudil Mesylate

99%+
A981488 现货 SPHINX31

SPHINX31 is a potent and selective inhibitor of serine/arginine-rich protein kinase 1 (SRPK1), with an IC50 of 5.9 nM. SPHINX31 inhibits phosphorylation of serine/arginine-rich splicing factor 1 (SRSF1). SPHINX31 is a potential topical therapeutic for neovascular eye disease[1].

99%+
A784195 现货 CMPD1

CMPD1 is a selective inhibitor of non-ATP-competitive p38 MAPK-mediated MK2 phosphorylation with apparent Ki (Kiapp) of 330 nM.

97%
A623292 现货 OSU-T315

ILK-IN-2 is a ILK inhibitor.

99%+
A569516 现货 GSK429286A

GSK429286A selectively inhibits ROCK1 and ROCK2 with the IC50 value of 14 nM and 63 nM, respectively.

99%+
A303159 现货 SAR407899

SAR407899 is a potent, ATP-competitive ROCK inhibitor woth Ki value of 36 nM/41 nM for human ROCK/Rat ROCK respectively.

99%+
A1218646 现货 SPHINX

99%+
A317869 现货 RKI-1447

RKI-1447 is a potent small molecule inhibitor of ROCK1 and ROCK2, with IC50 of 14.5 nM and 6.2 nM, respectively, and has anti-invasive and antitumor activities.

99%+
A119193 现货 Acteoside/类叶升麻苷

Acteoside, is a natural product isolated and purified from the herbs of Cistanche deserticola Y.C. Ma with known antioxidant activity. It is a protein kinase C inhibitor (IC50 =25 μM).

99%+
A1229590 现货 Nek2/Hec1-IN-2

98%+
A490626 现货 SRPIN340

SRPIN340 is an inhibitor of serine/arginine-rich protein kinase SRPK1 with IC50 of 0.89 μM.

99%+
Ambeed 相关网站 Ambeed.cn Ambeed.com
Ambeed
关于我们
联系我们
资讯中心
网站地图
产品手册
  • 批次文件查询
  • 客户支持
    专业术语
    缩略词释义
    质量手册
    产品咨询
    计算器
    活动政策
    订购方法
    活动声明
    联系我们
    400-920-2911 sales@ambeed.cn tech@ambeed.cn
    Ambeed 只为有资质的科研机构、医药企业基于科学研究或药证申报的用途提供医药研发服务,不为任何个人或者非科研性质用途提供服务。