A939572是一种强效且口服生物利用度的硬脂酰辅酶A去饱和酶1（SCD1）抑制剂，其对mSCD1和hSCD1的IC50值分别为<4 nM和37 nM。

XEN723 is a potent thiazolylimidazolidinone inhibitor of Stearoyl-CoA Desaturase (SCD1) with IC50s of 45 and 524 nM in mouse and HepG2 cell, respectively.

PluriSln 1 is an inhibitor of cell pluripotency and stearoyl-coA desaturase (SCD1) that can induce ER stress and apoptosis in hPSCs.

MF-438 is an inhibitor of stearoyl-CoA desaturase 1 (SCD1) with EC50 of 2.3 nM for rSCD1.

SCD1 inhibitor-4 is a potent and orally active SCD1 inhibitor.

MK-8245 is a liver-targeting inhibitor of stearoyl-CoA desaturase (SCD) with IC50 of 1 nM for human SCD1 and 3 nM for both rat SCD1 and mouse SCD1, with anti-diabetic and anti-dyslipidemic efficacy.

Aramchol is a conjugate of cholic acid and arachidic acid that could inhibit stearoyl coenzyme A desaturase 1 (SCD1) activity.

CVT-12012 is a potent and orally bioavailable stearoyl-coA desaturase (SCD) inhibitor, with IC50s of 38 nM, 6.1 nM for rat microsomal and human HEPG2, respectively.

SCD inhibitor 1 is an inhibitor of stearoyl-coa desaturase (SCD).