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货号 产品名 纯度
A809751 Mephenytoin

98%
A987492 Rhapontigenin 3'-O-glucoside/丹叶大黄素 3'-O-葡萄糖苷

98%
A1176909 4'-Methylchrysoeriol

99%+
A1721473 TP0472993

98%
A2248104 Opevesostat

Opevesostat是一种胆固醇侧链裂解酶(CYP11A1)的抑制剂。

95%
A252947 Polygalaxanthone III/远志山酮III

Polygalaxanthone III抑制CYP450酶,并抑制CYP2E1催化的chlorzoxazone 6-羟基化,其IC50为50.56μM。

99%
A1194181 7-Benzyloxy-4-(trifluoromethyl)coumarin

97%
A288033 Dihydromethysticin

Dihydromethysticin 是来自卡瓦(kava)的一种卡瓦内酯,诱导CYP3A23活性。

99%+
A465505 (±)-N-3-Benzylnirvanol/(+/-)-N-3-苄基神经醇

97%
A336445 1-Aminobenzotriazole/1-氨基苯并三唑

ABT is a non-specific cytochrome P450 (CYP) inhibitor.

95%
A696347 5-Bromo-2′-deoxy-2′-fluorouridine

98%
A508090 1-Ethynylnaphthalene/1-乙炔基萘

1-Ethynylnaphthalene is a selective inhibitor of cytochrome P450 1B1.

97%
A1325616 (E/Z)-DMU2105

DMU2105 is a potent CYP1B1 inhibitor with IC50 value of 10nM for human CYP1B1 enzyme bound to yeast-derived microsomes (Sacchrosomes™).

99%+
A676053 Methylsticin/麻醉椒苦素

97%
A399493 Orteronel

Orteronel is a highly selective inhibitor of human 17,20-lyase with IC50 of 38 nM, and exhibits > 1000-fold selectivity over other CYPs such as 11-hydroxylase and CYP3A4.

99%+
A133600 Bergaptol/香柑醇

Bergaptol 是一种抑制 CYP3A4 酶去甲基化活性的抑制剂,IC50 为 24.92 μM。最近的研究表明其具有抗增殖和抗癌特性。

98%
A435923 (S)-Mephenytoin

(S)-Mephenytoin is a substrate of the cytochrome P450 (CYP) isoform CYP2C19, also known as mephenytoin 4-hydroxylase.

99%+
A751790 4-Hydroxy-3,3-dimethylcyclohexanone

95+%
A767094 Curcumenol/莪术烯醇

Curcumenol inhibits NF-κB activation by suppressing the nuclear translocation of the NF-κB p65 subunit and blocking IκBα phosphorylation and degradation.

98%
A1228494 Mefentrifluconazole

Mefentrifluconazole is a novel azole derivative and used as an agrochemical broad-spectrum antifungal agent. Mefentrifluconazole is a potent, selective and orally active fungal CYP51 (Kd= 0.5 nM) inhibitor, but shows less inhibitory activity on human aromatase (IC50=0.92 μM).

98%
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