AR-C155858 是一种选择性单羧酸转运蛋白 MCT1 和 MCT2 的抑制剂，Ki 分别为 2.3 nM 和 10 nM。

7ACC2 is a potent MCT inhibitor with IC50 of 11 nM for inhibition of [14C]-lactate influx for antitumor treatment targeting lactate transport in cancer cells.

BAY-8002 is a potent MCT Inhibitor with IC50 value of 8nM for inhibition of L-lactate uptake.

AZD3965 is a potent, selective and orally available monocarboxylate transporter 1 (MCT1) inhibitor with a binding affinity of 1.6 nM.

α-Cyano-4-hydroxycinnamic acid is a MCT inhibitor with antitumoral and antiangiogenic activity.

7ACC1 selectively interfere with lactate fluxes in the lactate-rich tumor microenvironment and inhibits lactate influx but not efflux in tumor cells expressing MCT1 and MCT4 transporters.

UK-5099 is a potent is MPC (mitochondrial pyruvate carrier) inhibitor with IC50 value of 50 nM.

Silychristin, a natural product isolated and purified from the herbs of Silybum marianum (L.) Gaertn., is a plant growth regulator, an anti-hepatotoxic agent, and an inhibitor of horseradish peroxidases and lipoxygenase.

SR13800 is a cell-permeable inhibitor of monocarboxylate transporter 1 (MCT1).