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货号 产品名 纯度
A264157 现货 Talabostat mesylate

Talabostat mesylate (Val-boroPro mesylate; PT100 mesylate) 是一种口服活性、非选择性二肽基肽酶IV(DPP-IV)抑制剂(IC50 < 4 nM;Ki = 0.18 nM),也是首个临床上抑制成纤维细胞激活蛋白FAP)的抑制剂(IC50 = 560 nM)。它还抑制DPP8/9(IC50 = 4/11 nM;Ki = 1.5/0.76 nM)、静息细胞脯氨酸二肽酶(QPP)(IC50 = 310 nM)、DPP2其他DASH家族酶,表现出抗肿瘤和造血刺激活性。

98%+
A419052 现货 Saxagliptin hydrate/沙格列汀 水合物

Saxagliptin, the monohydrate form of anhydrous saxagliptin, is a reversible and selective DPP4 inhibitor with IC50 of 26 nM. It is used for the treatment of type 2 diabetes.

99%
A420160 现货 Alogliptin Benzoate/苯甲酸阿格列汀

Alogliptin benzoate is the benzoate salt form of alogliptin which is a selective inhibitor of DPP-4 with IC50 of 6.9 nM that exhibits greater selective than DPP-2, DPP-8 and DPP-9.

97%
A130556 现货 Saxagliptin hydrochloride/盐酸沙格列汀

Saxagliptin, also known as BMS-477118, is a new oral hypoglycemic (anti-diabetic drug) of the new dipeptidyl peptidase-4 (DPP-4) inhibitor class of drugs. Saxagliptin was approved in 2008 for the treatment of type 2 diabetes. Saxagliptin is a competitive DPP4 inhibitor that slows the inactivation of the incretin hormones, thereby increasing their bloodstream concentrations and reducing fasting and postprandial glucose concentrations in a glucose-dependent manner in patients with type 2 diabetes mellitus. .

98%
A323507 现货 Sitagliptin phosphate monohydrate/西他列汀磷酸盐一水合物

Sitagliptin Phosphate Monohydrate is a potent inhibitor of DPP4 with IC50 of 19 nM in Caco-2 cell extracts.

99%
A111654 现货 Sitagliptin phosphate/磷酸西他列汀

Sitagliptin phosphate is a potent inhibitor of DPP4 with IC50 of 19 nM in Caco-2 cell extracts.

98%
A850169 现货 DBPR108

DBPR108 is a potent, selective, and orally bioavailable dipeptide-derived inhibitor of DPP4 with IC50 of 15 nM showing no inhibition on DDP8 and DPP9.

98%+
A127061 现货 Sitagliptin/西格列汀

Sitagliptin is a potent inhibitor of DPP4 with IC50 of 19 nM in Caco-2 cell extracts.

98%
A392251 现货 Linagliptin/利拉利汀

Linagliptin, a purine and quinazoline derivative, can inhibit DPP-4 with IC50 of 1 nM. It functions as an incretin and is used as a hypoglycemic agents in the treatment of type 2 diabetes mellitus.

98%
A115550 现货 Omarigliptin/奥格列汀

Omarigliptin, also called MA-3102, is an selective inhibitor of DPP-4 with IC50 of 1.6 nM and Ki of 0.8 nM. Its selectivity is higher than other 168 proteasomes.

98%
A295732 现货 Alogliptin/阿格列汀

Alogliptin is a dipeptidyl peptidase 4 (DPP-4) inhibitor with IC50 of 6.9 nM that exhibits greater selective than DPP-2, DPP-8 and DPP-9.

98%
A354223 现货 Saxagliptin/沙格列汀

Saxagliptin is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.

98%
A253925 现货 Teneligliptin HBr/氢溴酸替格列汀

Teneligliptin Hydrobromide is a DPP4 inhibitor with IC50 value of <1 nM. It is commonly used as an add on treatment when meformin is not achieving the expected glycemic goals.

98%
A403832 现货 Vildagliptin/维达列汀

Vildagliptin is an inhibitor of DPP-4 with IC50 of 2.3 nM that is used in the treatment of type 2 diabetes mellitus.

98%
A114611 现货 Diprotin A

Diprotin A is the inhibitor of dipeptidyl peptidase IV. It can inhibit entry of HIV-1 or HIV-2 into T lymphoblastoid and monocytoid cell lines.

98%
A1210845 现货 NDMC101

NDMC101 is a potent osteoclastogenesis inhibitor and inhibits osteoclast differentiation via down-regulation of NFATc1-modulated gene express. NDMC101 is similar to the DPP4 substrate and is a significant inhibitor of early T-cell activation via DPP4 inhibition. NDMC101can be used for study of bone disorders, such as rheumatoid arthritis, and synovial inflammation et al .

99%+
A1163794 Prodipine HCl/普罗地平盐酸盐

99+%
A1176690 Diprotin A TFA

99+%
A165125 1G244

99%
A823508 Denagliptin

95+%
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