N-desmethyl Enzalutamide
产品说明书
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同义名 : | N-desmethyl MDV 3100 |
| CAS号 : | 1242137-16-1 | |
| 货号 : | A526563 | |
| 分子式 : | C20H14F4N4O2S | |
| 纯度 : | 99% | |
| 分子量 : | 450.41 | |
| MDL号 : | MFCD24386671 | |
| 存储条件： |
Pure form Sealed in dry,2-8°C In solvent -20°C:3-6个月-80°C:12个月 |
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| 溶解度 : |
DMSO: 105 mg/mL(233.12 mM)，配合低频超声助溶，注意：DMSO长时间开封后，会吸水并导致溶解能力下降，请避免使用长期开封的DMSO |
| 生物活性 | |||
|---|---|---|---|
| 描述 | N-desmethyl Enzalutamide is an active metabolite of Enzalutamide, demonstrating primary and secondary pharmacodynamics similar in potency to Enzalutamide itself. It circulates in plasma at concentrations comparable to those of Enzalutamide[1]. | ||
| 实验方案 | |||
|---|---|---|---|
| 1mg | 5mg | 10mg | |
|
1 mM 5 mM 10 mM |
2.22mL 0.44mL 0.22mL |
11.10mL 2.22mL 1.11mL |
22.20mL 4.44mL 2.22mL |
| 参考文献 |
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