WHI-P258
产品说明书
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同义名 : | - |
| CAS号 : | 21561-09-1 | |
| 货号 : | A480267 | |
| 分子式 : | C16H15N3O2 | |
| 纯度 : | 97% | |
| 分子量 : | 281.31 | |
| MDL号 : | MFCD01815294 | |
| 存储条件： |
Pure form Keep in dark place, sealed in dry, store in freezer, under -20°C In solvent -20°C:3-6个月-80°C:12个月 |
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| 溶解度 : |
DMSO: 30 mg/mL(106.64 mM)，配合低频超声助溶，注意：DMSO长时间开封后，会吸水并导致溶解能力下降，请避免使用长期开封的DMSO |
| 生物活性 | |||
|---|---|---|---|
| 描述 | WHI-P258 is a quinazoline compound that binds to the active site of JAK3 with an estimated Ki value of 72 µM. WHI-P258 does not inhibit JAK3 and does not affect thrombin-induced platelet aggregation even at a concentration of 100 µM[1][2]. | ||
| 实验方案 | |||
|---|---|---|---|
| 1mg | 5mg | 10mg | |
|
1 mM 5 mM 10 mM |
3.55mL 0.71mL 0.36mL |
17.77mL 3.55mL 1.78mL |
35.55mL 7.11mL 3.55mL |
| 参考文献 |
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