Istaroxime

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Chemical Structure| 203737-93-3 同义名 : PST2744
CAS号 : 203737-93-3
货号 : A352208
分子式 : C21H32N2O3
纯度 : 99+%
分子量 : 360.49
MDL号 : N/A
存储条件：

Pure form

In solvent -20°C:3-6个月-80°C:12个月
溶解度 : -
生物活性
描述 Istaroxime is a potent inhibitor of Na+,K+-ATPase with IC50 of 0.11 μM.
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

2.77mL

0.55mL

0.28mL

13.87mL

2.77mL

1.39mL

27.74mL

5.55mL

2.77mL
参考文献

[1]Gobbini M, Armaroli S, et al. Novel analogues of Istaroxime, a potent inhibitor of Na(+),K(+)-ATPase: Synthesis, structure-activity relationship and 3D-quantitative structure-activity relationship of derivatives at position 6 on the androstane scaffold. Bioorg Med Chem. 2010 Jun 15;18(12):4275-99.

[2]Gobbini M, Armaroli S, et al. Novel analogues of istaroxime, a potent inhibitor of Na+,K+-ATPase: synthesis and structure-activity relationship. J Med Chem. 2008 Aug 14;51(15):4601-8.