FAAH-IN-2
产品说明书
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同义名 : | - |
| CAS号 : | 184475-71-6 | |
| 货号 : | A207764 | |
| 分子式 : | C15H11ClFN3O2 | |
| 纯度 : | 98% | |
| 分子量 : | 319.72 | |
| MDL号 : | MFCD09908046 | |
| 存储条件： |
Pure form Keep in dark place, inert atmosphere, store in freezer, under -20°C In solvent -20°C:3-6个月-80°C:12个月 |
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| 溶解度 : |
DMSO: 20 mg/mL(62.56 mM)，配合低频超声助溶，注意：DMSO长时间开封后，会吸水并导致溶解能力下降，请避免使用长期开封的DMSO |
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| 动物实验配方： |
| 生物活性 | |||
|---|---|---|---|
| 描述 | Fatty acid amide hydrolase (FAAH), an integral membrane bound enzyme and a member of the extensive family of serine hydrolases referred to as amidase signature (AS) family, catalyses degradation of lipid signalling fatty acid amides including the sleep-inducing oleamide and endogenous cannabinoid anandamide (AEA)[2]. FAAH-IN-2 (O-Desmorpholinopropyl Gefitinib), a metabolite of Gefitinib, is a potent FAAH inhibitor. | ||
| 实验方案 | |||
|---|---|---|---|
| 1mg | 5mg | 10mg | |
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1 mM 5 mM 10 mM |
3.13mL 0.63mL 0.31mL |
15.64mL 3.13mL 1.56mL |
31.28mL 6.26mL 3.13mL |
| 参考文献 |
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