CBP/p300-IN-3

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Chemical Structure| 2299226-01-8 同义名 : -
CAS号 : 2299226-01-8
货号 : A1365010
分子式 : C24H29N7O
纯度 : 99%
分子量 : 431.53
MDL号 : MFCD32201113
存储条件：

Pure form Sealed in dry, 2-8°C

In solvent -20°C:3-6个月-80°C:12个月
溶解度 :

DMSO: 250 mg/mL(579.33 mM)，配合低频超声助溶，注意：DMSO长时间开封后，会吸水并导致溶解能力下降，请避免使用长期开封的DMSO
生物活性
描述 CBP/p300-IN-3 is a histone acetyltransferase inhibitor targeting p300/CBP. It originates from patent WO 2019049061 A1[1].
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

2.32mL

0.46mL

0.23mL

11.59mL

2.32mL

1.16mL

23.17mL

4.63mL

2.32mL
参考文献

[1]Medina, et al. 5-(1H-Benzo[d]imidazol-2-yl)pyridin-2-amine and 5-(3H-imidazo[4,5-b]pyridin-6-yl)pyridin-2-amine derivatives as c-MYC and p300/CBP histone acetyltransferase inhibitors for treating cancer and their preparation.