| 生物活性 | |||
|---|---|---|---|
| 靶点 | 
 | ||
| 描述 | PUN51207 is a CK1 inhibitor with IC50 values of 15nM and 16nM for CK1δ and CK1ε, respectively, as well as exhibits inhibitory effect on p38α MAPK with IC50 value of 73nM. | ||
| 实验方案 | |||
|---|---|---|---|
| 1mg | 5mg | 10mg | |
| 1 mM 5 mM 10 mM | 2.61mL 0.52mL 0.26mL | 13.04mL 2.61mL 1.30mL | 26.08mL 5.22mL 2.61mL | 
| 参考文献 | 
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