GSK2193874 is a selective transient receptor potential vanilloid 4 (TRPV4) blocker with IC50 value of 0.04 μM.
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Type
HazMat fee for 500 gram (Estimated)
Excepted Quantity
USD 0.00
Limited Quantity
USD 15-60
Inaccessible (Haz class 6.1), Domestic
USD 80+
Inaccessible (Haz class 6.1), International
USD 150+
Accessible (Haz class 3, 4, 5 or 8), Domestic
USD 100+
Accessible (Haz class 3, 4, 5 or 8), International
GSK2193874 is an orally administered, highly potent, and selective antagonist of TRPV4, demonstrating IC50 values of 2 nM for rTRPV4 and 40 nM for hTRPV4. When tested against various TRP channels, GSK2193874 shows selectivity, with no significant activity against TRPV1, TRPA1, TRPC3, TRPC6, and TRPM8, all having IC50 values greater than 25 μM[1].
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