生物活性 | |||
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描述 | CP94253 HCl is a potent and selective agonist of the 5-HT1B receptor with a Ki value of 2 nM. the Ki values for the 5-HT1A, 5-HT1D, 5-HT1C, and 5-HT2 receptors are 89, 49, 860, and 1600 nM, respectively[1] . CP94253 HCl is centrally active when administered systemically in vivo[2].CP94253 HCl is centrally active when administered systemically in vivo [2]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
3.40mL 0.68mL 0.34mL |
17.02mL 3.40mL 1.70mL |
34.04mL 6.81mL 3.40mL |