CP94253 HCl

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Chemical Structure| 845861-39-4 同义名 : CP 94,253 (hydrochloride); CP94253 hydrochloride
CAS号 : 845861-39-4
货号 : A798375
分子式 : C15H20ClN3O
纯度 : 99%+
分子量 : 293.79
MDL号 : MFCD03453293
存储条件:

Pure form Sealed in dry,Store in freezer, under -20°C

In solvent -20°C:3-6个月-80°C:12个月

溶解度 : -
动物实验配方:
生物活性
描述 CP94253 HCl is a potent and selective agonist of the 5-HT1B receptor with a Ki value of 2 nM. the Ki values for the 5-HT1A, 5-HT1D, 5-HT1C, and 5-HT2 receptors are 89, 49, 860, and 1600 nM, respectively[1] . CP94253 HCl is centrally active when administered systemically in vivo[2].CP94253 HCl is centrally active when administered systemically in vivo [2].
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

3.40mL

0.68mL

0.34mL

17.02mL

3.40mL

1.70mL

34.04mL

6.81mL

3.40mL