Bromopride

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Chemical Structure| 4093-35-0 同义名 : 溴灭吐灵 ;Emepride; Viadil; Emoril
CAS号 : 4093-35-0
货号 : A764267
分子式 : C14H22BrN3O2
纯度 : 99%
分子量 : 344.25
MDL号 : N/A
存储条件:

Pure form Keep in dark place, inert atmosphere, 2-8°C

In solvent -20°C:3-6个月-80°C:12个月

溶解度 : -
动物实验配方:
生物活性
描述 Bromopride is a dopamine antagonist with prokinetic properties, widely used as an antiemetic.
临床研究
NCT号 适应症或疾病 临床期 招募状态 预计完成时间 地点
NCT02604576 Dyspepsia Phase 3 Recruiting August 2018 Brazil ... 展开 >> Centro de Medicina Reprodutiva Carlos Isaia Filho Ltda Recruiting Porto Alegre, Rio Grande Do Sul, Brazil Contact: Carlos Isaia Filho, MD          Hospital de Clínicas de Porto Alegre Recruiting Porto Alegre, Rio Grande Do Sul, Brazil Contact: Carlos Fernando Francesconi, MD          Hospital Ernesto Dornelles Recruiting Porto Alegre, RS, Brazil, 90160-092 Contact: Guilherme B. Sander, MD          UNIFAG Recruiting Bragança Paulista, SP, Brazil, 129169000 Contact: José Pedrazzoli, MD          Loema Recruiting Campinas, SP, Brazil, 13010001 Contact: Fabio R Santos, MD       contato@loemaipc.com.br    Principal Investigator: Fabio R Santos, MD          Instituto de Pesquisa Clinica de Campinas Recruiting Campinas, SP, Brazil, 13060-080 Contact: José Francisco K. Saraiva, MD          Centro de Estudos Clínicos do Interior Paulista Recruiting Jau, SP, Brazil, 17201-130 Contact: Paula Tokunaga, MD          Faculdade de Medicina do ABC Recruiting Santo André, SP, Brazil, 09060-650 Contact: Wilson Catapani, MD          AFIP Recruiting São Paulo, Sâo Paulo, Brazil, 04020-060 Contact: Edson Ide, MD          Allergisa Recruiting Campinas, São Paulo, Brazil Contact: Mauro A Crippa, MD 收起 <<
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

2.90mL

0.58mL

0.29mL

14.52mL

2.90mL

1.45mL

29.05mL

5.81mL

2.90mL

参考文献

[1]Silva SM, Jerônimo MS, et al. Effects of bromopride on expression of metalloproteinases and interleukins in left colonic anastomoses: an experimental study. Braz J Med Biol Res. 2014 Oct;47(10):911-6.

[2]Marques e Silva S, Ferreira VM, et al. Effects of bromopride on the healing of left colon anastomoses of rats. Rev Col Bras Cir. 2011 Nov-Dec;38(6):429-34. English, Portuguese.