BMS-986158
产品说明书
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同义名 : | - |
| CAS号 : | 1800340-40-2 | |
| 货号 : | A723935 | |
| 分子式 : | C30H33N5O2 | |
| 纯度 : | 99%+ | |
| 分子量 : | 495.62 | |
| MDL号 : | MFCD31544327 | |
| 存储条件： |
Pure form Sealed in dry, room temperature In solvent -20°C:3-6个月-80°C:12个月 |
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| 溶解度 : | - | |
| 动物实验配方： |
| 生物活性 | |||
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| 靶点 |
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| 描述 | BMS-986158 is an effective BET inhibitor, with IC50 values of 6.6 nM in NCI-H211 small cell lung cancer (SCLC) cells and 5 nM in MDA-MB231 triple-negative breast cancer (TNBC) cells[1]. | ||
| 实验方案 | |||
|---|---|---|---|
| 1mg | 5mg | 10mg | |
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1 mM 5 mM 10 mM |
2.02mL 0.40mL 0.20mL |
10.09mL 2.02mL 1.01mL |
20.18mL 4.04mL 2.02mL |
