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同义名 : | - |
CAS号 : | 152239-46-8 | |
货号 : | A601317 | |
分子式 : | C14H14N4OS | |
纯度 : | 99%+ | |
分子量 : | 286.35 | |
MDL号 : | MFCD00923644 | |
存储条件: |
Pure form Sealed in dry, 2-8°C In solvent -20°C:3-6个月-80°C:12个月 |
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溶解度 : | - | |
动物实验配方: |
生物活性 | |||
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描述 | SB 204741 is a selective high-affinity 5-HT2B antagonist with a pKi value of 7.1. SB 204741 is approximately 20-fold more selective for human 5-HT2B receptors than for human 5-HT2C receptors [1]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
3.49mL 0.70mL 0.35mL |
17.46mL 3.49mL 1.75mL |
34.92mL 6.98mL 3.49mL |