Rilapladib

产品说明书

Print
Chemical Structure| 412950-08-4 同义名 : SB 659032
CAS号 : 412950-08-4
货号 : A534662
分子式 : C40H38F5N3O3S
纯度 : 99%
分子量 : 735.81
MDL号 : MFCD13195581
存储条件：

Pure form Sealed in dry, store in freezer, under -20°C

In solvent -20°C:3-6个月-80°C:12个月
溶解度 : -
动物实验配方：
生物活性
描述 SB-659032 is a selective and orally active inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) that is being developed for the treatment of atherosclerosis.
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

1.36mL

0.27mL

0.14mL

6.80mL

1.36mL

0.68mL

13.59mL

2.72mL

1.36mL
参考文献

[1]Tawakol A, Singh P, et al. Effect of treatment for 12 weeks with rilapladib, a lipoprotein-associated phospholipase A2 inhibitor, on arterial inflammation as assessed with 18F-fluorodeoxyglucose-positron emission tomography imaging. J Am Coll Cardiol. 2014 Jan 7-14;63(1):86-8.