FN-1501

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Chemical Structure| 1429515-59-2 同义名 : -
CAS号 : 1429515-59-2
货号 : A512950
分子式 : C22H25N9O
纯度 : 97%
分子量 : 431.49
MDL号 : MFCD31657383
存储条件:

Pure form Keep in dark place, sealed in dry, 2-8°C

In solvent -20°C:3-6个月-80°C:12个月

溶解度 : -
动物实验配方:
生物活性
描述 FN-1501 is a potent inhibitor of FLT3 and CDK, with IC50s of 2.47, 0.85, 1.96, and 0.28 nM for CDK2/cyclin A, CDK4/cyclin D1, CDK6/cyclin D1 and FLT3, respectively; has anticancer activity.
临床研究
NCT号 适应症或疾病 临床期 招募状态 预计完成时间 地点
NCT03690154 Advanced Cancer ... 展开 >> Solid Tumor 收起 << Phase 1 Recruiting August 2019 United States, Kansas ... 展开 >> KUMC Cancer Center Recruiting Fairway, Kansas, United States, 66205 Contact: Stephen K Williamson, MD    913-945-5059    swilliam@kumc.edu    Principal Investigator: Stephen K Williamson, MD          United States, Michigan Karmanos Cancer Institute Recruiting Detroit, Michigan, United States, 48334 Contact: Ulka Vaishampayan, MD    248-538-4701    vaishamu@karmanos.org    Principal Investigator: Ulka Vaishampayan, MD          Australia, Victoria Cabrini Malvern Hospital Recruiting Malvern, Victoria, Australia, 3144 Contact: Gary E Richardson, MD    1 300-300-977    gary.richardson@ocv.net.au    Principal Investigator: Gary E Richardson, MD 收起 <<
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

2.32mL

0.46mL

0.23mL

11.59mL

2.32mL

1.16mL

23.18mL

4.64mL

2.32mL