MK-5046

产品说明书

Print
Chemical Structure| 1022152-70-0 同义名 : -
CAS号 : 1022152-70-0
货号 : A384091
分子式 : C20H18F6N4O
纯度 : 98%
分子量 : 444.37
MDL号 : MFCD18782708
存储条件：

Pure form Sealed in dry, room temperature

In solvent -20°C:3-6个月-80°C:12个月
溶解度 : -
动物实验配方：
生物活性
描述 MK-5046 is a BRS-3 agonist, binds to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

2.25mL

0.45mL

0.23mL

11.25mL

2.25mL

1.13mL

22.50mL

4.50mL

2.25mL
参考文献

[1]Guan XM, et al. Antiobesity effect of MK-5046, a novel bombesin receptor subtype-3 agonist. J Pharmacol Exp Ther. 2011 Feb;336(2):356-364.