Gabazine

产品说明书

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Chemical Structure| 104104-50-9 同义名 : SR 95531 (hydrobromide); SR95531
CAS号 : 104104-50-9
货号 : A283069
分子式 : C15H18BrN3O3
纯度 : 95+%
分子量 : 368.23
MDL号 : MFCD09055424
存储条件：

Pure form Sealed in dry,2-8°C

In solvent -20°C:3-6个月-80°C:12个月
溶解度 : -
动物实验配方：
生物活性
描述 Gabazine hydrobromide is a drug that acts as an antagonist at GABAA receptors. It is used in scientific research and has no role in medicine, as it would be expected to produce convulsions if used in humans.
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

2.72mL

0.54mL

0.27mL

13.58mL

2.72mL

1.36mL

27.16mL

5.43mL

2.72mL
参考文献

[1]Arguedas AG, Akaniro JC, et al. In vitro activity of tosufloxacin, a new quinolone, against respiratory pathogens derived from cystic fibrosis sputum. Antimicrob Agents Chemother. 1990 Nov;34(11):2223-7.

[2]Ueno S, Bracamontes J, et al. Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA receptor. J Neurosci. 1997 Jan 15;17(2):625-34.