Tie2 kinase inhibitor 1
产品说明书
 |
同义名 : | Tunica Interna Endothelial Cell Kinase 2 Inhibitor; Tie2 Kinase Inhibitor; Compound 5; Tie2 kinase inhibitor 5; Tie2 inhibitor 5; Tie2-IN-5 |
| CAS号 : | 948557-43-5 | |
| 货号 : | A253059 | |
| 分子式 : | C26H21N3O2S | |
| 纯度 : | 99%+ | |
| 分子量 : | 439.53 | |
| MDL号 : | MFCD18384977 | |
| 存储条件： |
Pure form Keep in dark place, sealed in dry, 2-8°C In solvent -20°C:3-6个月-80°C:12个月 |
|
| 溶解度 : | - | |
| 动物实验配方： |
| 生物活性 | |||
|---|---|---|---|
| 靶点 |
|
||
| 描述 | Tie2 kinase inhibitor 1 is a strong and selective inhibitor of Tie2 kinase, exhibiting an IC50 value of 250 nM. It has shown an IC50 of 50 μM against p38 and demonstrates moderate to high efficacy in cellular assays, with a cellular IC50 of 232 nM[1]. It exhibits anti-cancer properties[2]. | ||
| 实验方案 | |||
|---|---|---|---|
| 1mg | 5mg | 10mg | |
|
1 mM 5 mM 10 mM |
2.28mL 0.46mL 0.23mL |
11.38mL 2.28mL 1.14mL |
22.75mL 4.55mL 2.28mL |
