L-NMMA acetate

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Chemical Structure| 53308-83-1 同义名 : Tilarginine acetate; Methylarginine acetate; NG-Monomethyl-L-arginine acetate; ANO-1020; L-NG-monomethyl Arginine acetate; L-NMMA (acetate)
CAS号 : 53308-83-1
货号 : A177581
分子式 : C9H20N4O4
纯度 : 98%
分子量 : 248.28
MDL号 : MFCD00069311
存储条件:

Pure form Sealed in dry,2-8°C

In solvent -20°C:3-6个月-80°C:12个月

溶解度 : -
动物实验配方:
生物活性
描述 L-NMMA acetate is a nitric oxide synthase inhibitor of all NOS isoforms including NOS1, NOS2, and NOS3. The Ki values for nNOS (rat), eNOS (human), and iNOS (mouse) are approximately 0.18, 0.4, and 6 µM, respectively.
临床研究
NCT号 适应症或疾病 临床期 招募状态 预计完成时间 地点
NCT00112281 Shock, Cardiogenic Phase 3 Terminated - -
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

4.03mL

0.81mL

0.40mL

20.14mL

4.03mL

2.01mL

40.28mL

8.06mL

4.03mL