G36
产品说明书
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同义名 : | - |
| CAS号 : | 1392487-51-2 | |
| 货号 : | A1339164 | |
| 分子式 : | C22H22BrNO2 | |
| 纯度 : | 99%+ | |
| 分子量 : | 412.32 | |
| MDL号 : | MFCD28137712 | |
| 存储条件： |
Pure form Sealed in dry, store in freezer, under -20°C In solvent -20°C:3-6个月-80°C:12个月 |
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| 溶解度 : | - | |
| 动物实验配方： |
| 生物活性 | |||
|---|---|---|---|
| 描述 | G36 is a cell-permeable, non-steroidal G protein-coupled estrogen receptor (GPER/GPR30) antagonist that selectively inhibits estrogen-mediated activation of PI3K by GPER but not by ERα. G36 also inhibits estrogen-mediated calcium mobilization(IC50=112 nM)[1]. | ||
| 实验方案 | |||
|---|---|---|---|
| 1mg | 5mg | 10mg | |
|
1 mM 5 mM 10 mM |
2.43mL 0.49mL 0.24mL |
12.13mL 2.43mL 1.21mL |
24.25mL 4.85mL 2.43mL |
