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同义名 : | EPI-506 |
CAS号 : | 1637573-04-6 | |
货号 : | A1275527 | |
分子式 : | C27H33ClO8 | |
纯度 : | 97% | |
分子量 : | 521.0 | |
MDL号 : | N/A | |
存储条件: |
Pure form Sealed in dry, 2-8°C In solvent -20°C:3-6个月-80°C:12个月 |
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溶解度 : | - | |
动物实验配方: |
生物活性 | |||
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描述 | Ralaniten triacetate (EPI-506), a precursor of Ralaniten, is the first orally active inhibitor targeting the androgen receptor (AR) N-terminal domain (NTD). It is effective against both the full-length AR and variants associated with resistance, such as AR-v7[1][2]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
1.92mL 0.38mL 0.19mL |
9.60mL 1.92mL 0.96mL |
19.19mL 3.84mL 1.92mL |
参考文献 |
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