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同义名 : | PF-06685360 |
CAS号 : | 1527475-61-1 | |
货号 : | A1177088 | |
分子式 : | C16H16N6O | |
纯度 : | 98% | |
分子量 : | 308.34 | |
MDL号 : | MFCD31697701 | |
存储条件: |
Pure form Sealed in dry, 2-8°C In solvent -20°C:3-6个月-80°C:12个月 |
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溶解度 : | - | |
动物实验配方: |
生物活性 | |||
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描述 | PFE-360 , also known as PF-06685360, is a potent, selective, brain-penetrating and orally active LRRK2 inhibitor with an in vivo mean IC50 value of 2.3 nM[1][2]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
3.24mL 0.65mL 0.32mL |
16.22mL 3.24mL 1.62mL |
32.43mL 6.49mL 3.24mL |