PFE-360

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Chemical Structure| 1527475-61-1 同义名 : PF-06685360
CAS号 : 1527475-61-1
货号 : A1177088
分子式 : C16H16N6O
纯度 : 98%
分子量 : 308.34
MDL号 : MFCD31697701
存储条件:

Pure form Sealed in dry, 2-8°C

In solvent -20°C:3-6个月-80°C:12个月

溶解度 : -
动物实验配方:
生物活性
描述 PFE-360 , also known as PF-06685360, is a potent, selective, brain-penetrating and orally active LRRK2 inhibitor with an in vivo mean IC50 value of 2.3 nM[1][2].
实验方案
1mg 5mg 10mg

1 mM

5 mM

10 mM

3.24mL

0.65mL

0.32mL

16.22mL

3.24mL

1.62mL

32.43mL

6.49mL

3.24mL