Mizacorat
产品说明书
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同义名 : | AZD9567 |
| CAS号 : | 1893415-00-3 | |
| 货号 : | A1177085 | |
| 分子式 : | C27H28F2N4O3 | |
| 纯度 : | 99%+ | |
| 分子量 : | 494.53 | |
| MDL号 : | MFCD31619227 | |
| 存储条件： |
Pure form Sealed in dry, 2-8°C In solvent -20°C:3-6个月-80°C:12个月 |
|
| 溶解度 : | - | |
| 动物实验配方： |
| 生物活性 | |||
|---|---|---|---|
| 描述 | Mizacorat is a potent, orally active, non-steroidal and selective glucocorticoid receptor modulator (SGRM) with an IC50 of 3.8 nM. It has demonstrated superior efficacy in a streptococcal cell wall (SCW) reactivation model of joint inflammation[1]. | ||
| 实验方案 | |||
|---|---|---|---|
| 1mg | 5mg | 10mg | |
|
1 mM 5 mM 10 mM |
2.02mL 0.40mL 0.20mL |
10.11mL 2.02mL 1.01mL |
20.22mL 4.04mL 2.02mL |
