Dafadine-A, an analog of dafadine, is an inhibitor of DAF-9 cytochrome P450 in the nematode Caenorhabditis elegans and also inhibits the mammalian ortholog of DAF-9 (CYP27A1).

ABT is a non-specific cytochrome P450 (CYP) inhibitor.

Proadifen HCl is a nonspecific cytochrome P450 inhibitor, it's also a noncompetitive inhibitor of acetylcholine nicotinic receptors with IC50 of 19 μM in mouse skeletal muscle.

Uniconazole inhibits CK biosynthesis by suppressing CYP735A activity in Arabidopsis. Uniconazole inhibits the biosynthesis of gibberellin (GA), and brassinosteroid (BR) and the catabolism of abscisic acid (ABA).

1-Ethynylnaphthalene is a selective inhibitor of cytochrome P450 1B1.

DMU2105 is a potent CYP1B1 inhibitor with IC50 value of 10nM for human CYP1B1 enzyme bound to yeast-derived microsomes (Sacchrosomes™).

Furafylline is a potent and selective inhibitor of human cytochrome P450IA2 with IC50 of 0.07 μM.

Bergaptin is a competitive inhibitor of CYP1A1 with Ki of 10.7 nM.

(S)-Mephenytoin is a substrate of the cytochrome P450 (CYP) isoform CYP2C19, also known as mephenytoin 4-hydroxylase.

Cecropin B can inhibit the expression of CYP3A29.

Mefentrifluconazole is a novel azole derivative and used as an agrochemical broad-spectrum antifungal agent. Mefentrifluconazole is a potent, selective and orally active fungal CYP51 (Kd= 0.5 nM) inhibitor, but shows less inhibitory activity on human aromatase (IC50=0.92 μM).

Oteseconazole is a tetrazole antifungal agent potentially for the treatment of candidal vaginal infection by inhibiting sterol 14α-demethylase (CYP51).

NTP42 is a TxA2 Synthetase antagonist with IC50 value of 3.278nM.

Flavone can effect CYP (P450) activity, it's a class of flavonoids with antioxidant, anti-proliferative, anti-tumor, anti-microbial, estrogenic, acetyl cholinesterase, anti-inflammatory activities and are also used in cancer, cardiovascular disease, neurodegenerative disorders etc.

Dazoxiben hydrochloride is a potent, orally active thromboxane (TX) synthase inhibitor that reduces the formation of blood clots.

5-Methoxypsoralen, a naturally occurring linear furocoumarin, has been successfully used in combination with ultraviolet (UV) A irradiation [psoralen plus UV (PUVA)] to manage psoriasis and vitiligo and inhibits proliferation in the human hepatocellular carcinoma cell line.

Ramatroban is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.

Metyrapone is an inhibitor of cytochrome P450-mediated ω/ω-1 hydroxylase activity and CYP11B1.

Benzbromarone is a CYP2C9 inhibitor with Ki of 19.3 nM.