Litronesib is a selective, allosteric inhibitor of Eg5, which may result in mitotic disruption, apoptosis and consequently cell death in tumor cells that are actively dividing.

Kif15-IN-1 is a potent Kif15 kinesin inhibitor and inhibits cellular proliferation in tumor cell lines.

GSK923295 is a specific allosteric CENP-E inhibito with Ki value of 3.2 nM.

SB-743921 is a potent KIF11 inhibitor with Ki value of 0.1 nM.

Monastrol is a specific and allosteric inhibitor of mitotic molecular motor kinesin Eg5 with IC50 value of 14 μM.

BRD9876 is a selective inhibitor of MM1S growth. It is selective for microtubule bound Eg5 and causes a rapid arrest in G2/M phase.

Ispinesib is a quinazolinone-derived, specific and reversible kinesin spindle protein inhibitor with Ki_app value of 1.7 nM.

AZ3146 is a selective and potent Mps1 inhibitor with IC50 value of 35 nM.

MPI-0479605 is a potent and selective ATP competitive Mps1 with IC50 value of 1.8 nM.

H-Cys(Trt)-OH is a potent and selective inhibitor of mitotic kinesin Eg5 with IC50 value of 140 nM.