Gabazine hydrobromide is a drug that acts as an antagonist at GABAA receptors. It is used in scientific research and has no role in medicine, as it would be expected to produce convulsions if used in humans.

Broflanilide is a potential insecticide and metabolized to desmethyl-broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin (RDL) GABA receptor, and inhibits S. litura RDL GABAR, with an IC50 value of 1.3 nM.

CL 218872 is an agonist of benzodiazepine which displaying selectivity for α1 subunit-containing GABAA receptors with Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 nM for α1, α2, α3, α4, α5 and α6-subunit containing receptors respectively.

Etifoxine is potentiator of GABAA receptor function in cultured neurons.

AZD-7325 is a GABA-Aα2,3 selective receptor modulator.

NS11394 is a potent and subtype-selective GABA (A) receptor-positive modulator, possessing a functional efficacy selectivity profile of alpha(5) > alpha(3) > alpha(2) > alpha(1) at GABA (A) alpha subunit-containing receptors.

AWD 131-138 is a partial agonist of benzodiazepine receptor with effective anticonvulsant and anxiolytic properties.

Basmisanil is a selective modulator of GABAAα5 with negative allosteric regulation.

Loreclezole is a subtype-selective GABAA receptor modulator. Acts as a positive allosteric modulator of β2 or β3-subunit containing receptors.

U93631 is a ligand of GABAA receptor ligand (IC50 = 100 nM) which can induce a rapid decay of GABA-induced chloride currents.

L-655708 is a potent α5 subunit-selective GABAA receptor inverse agonist (Ki = 0.45 nM).

Gabapentin is a GABA analogue, used to treat seizures and neuropathic pain.

SAGE-217 is an agonist of GABAA receptor with EC50s of 296 nM and 163 nM for α1β2γ2 and α4β3δ respectively.

Tiagabine HCl is an inhibitor of gamma-aminobutyric acid (GABA) reuptake (IC50 = 67 nM in vivo) with anticonvulsant effect.

Ocinaplon is a modulator of GABAA receptors with anxiolytic activity. It displays modest selectivity for GABAA α1 receptors and partial agonist activity at α2-, α3- and α5-containing receptors.

Phytol can activite PPARα and attenuate the inflammatory response by inhibiting neutrophil migration and oxidative stress. Phytol is isolated from the leaves of black tea and acts as an aromatic ingredient.

L-cycloserine is an inhibitor of serine palmitoyltransferase and block sphingosine biosynthesis. It has antibiotic effective against mycobacterium tuberculosis.

Isoguvacine hydrochloride is a specific agonist of GABAA receptor.