LY2183240 is a highly potent blocker of anandamide uptake (IC50 = 270 pM).

JNJ-1661010 is a selective inhibitor of FAAH with IC50 of 10 nM (rat) and 12 nM (human).

URB937 is a FAAH inhibitor and increases anandamide levels, with an IC50 of 26.8 nM. URB937 fails to affect FAAH activity in the brain .

FAAH inhibitor 1 is a potent fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 18±8 nM.

Macamide B is a natural product isolated and purified from the herbs of Lepidium meyenii Walp.

Luminol is a chemical with chemiluminescence property, soluble in most polar organic solvents, insoluble in water. When mixed with an appropriate oxidizing agent, it emits a blue glow.

PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.

PF-04457845 selectively inhibits FAAH with an IC50 of 7.2 nM. It has anti-inflammatory effects and is used as analgesic.

URB-597 is fatty acid amide hydrolase (FAAH, IC50 = 4.6 nM) inhibitor without effect on other cannabinoid-related targets.

PF-750 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor with IC50 of 16.2 nM.

JZL195 functions as a dual inhibitor of FAAH and MAGL with IC50 of 13 nM and 19 nM respectively in brain of mouse.

Biochanin A, a phytoestrogen from Trifolium pratense, is an inhibitor of PTK with IC50 of 91.5 μM. It also can be metabolized in vivo to genistein.

BIA10-2474 is an inhibitor of fatty acid amide hydrolase (FAAH) with IC50 of 4.9 nM.